SCHEMBL10138488

SCHEMBL10138488

Bc1ccc(OCC)c(OCC)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 2/20 0.40
ALDH1A1 P00352 8/20 0.39
KDM4E B2RXH2 8/20 0.39
L3MBTL1 Q9Y468 4/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2D6 P10635 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KDM1A O60341 2/20 0.36
HSD17B10 Q99714 4/20 0.36
HPGD P15428 2/20 0.36
MAPT P10636 3/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NQO1 P15559 1/20 0.34
TSHR P16473 1/20 0.34
GAA P10253 1/20 0.34
MAPK1 P28482 2/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801007 0.88 KDM1A (0.41) TUBB1ALDH1A1KDM4EL3MBTL1CYP1A2
SCHEMBL13140816 0.81 TSHR (0.36) TUBB1ALDH1A1KDM4EL3MBTL1CYP1A2
SCHEMBL2123778 0.80 TUBB1 (0.40) TUBB1ALDH1A1KDM4EL3MBTL1CYP1A2
SCHEMBL14190820 0.80 ALDH1A1 (0.44) TUBB1ALDH1A1KDM4EL3MBTL1CYP1A2
SCHEMBL10909552 0.78 ALDH1A1 (0.48) TUBB1ALDH1A1KDM4EL3MBTL1CYP1A2
SCHEMBL17527769 0.78 L3MBTL1 (0.48) TUBB1ALDH1A1KDM4EL3MBTL1CYP1A2
SCHEMBL9196941 0.78 ALDH1A1 (0.48) TUBB1ALDH1A1KDM4EL3MBTL1HSD17B10
SCHEMBL27634810 0.76 ALDH1A1 (0.41) TUBB1ALDH1A1KDM4EL3MBTL1CYP1A2
SCHEMBL12645303 0.74 TSHR (0.41) TUBB1ALDH1A1L3MBTL1HSD17B10TSHR
SCHEMBL5042606 0.74 LMNA (0.45) TUBB1ALDH1A1KDM4EL3MBTL1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2444393-A1 Methods for producing cyclic benzamidine derivatives Eisai R&D Management Co., Ltd. (JP) 2012-04-25 EP disclosed
US-7375236-B2 Methods for producing cyclic benzamidine derivatives EISAI CO., LTD. (JP) 2008-05-20 US disclosed