SCHEMBL10144287

SCHEMBL10144287

Cc1cc(F)ccc1CN1C(=N)N[C@](CCC2CCCCC2)(CC2CCCCC2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
SLC6A4 P31645 2/20 0.36
KMT2A Q03164 2/20 0.35
BACE1 P56817 6/20 0.34
CTSD P07339 1/20 0.34
OPRL1 P41146 3/20 0.33
P2RX7 Q99572 2/20 0.32
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
TRPC5 Q9UL62 1/20 0.32
BCHE P06276 1/20 0.31
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7510721 0.89 ALDH1A1 (0.39) HTR2AHTR2CSLC6A4KMT2AP2RX7
SCHEMBL13613821 0.89 OPRM1 (0.36) KMT2ABACE1CTSDOPRL1P2RX7
SCHEMBL7512649 0.86 KMT2A (0.37) KMT2ABACE1CTSDMEN1ALDH1A1
SCHEMBL7512656 0.84 ALDH1A1 (0.46) KMT2ABACE1CTSDMEN1RAB9A
SCHEMBL7510402 0.82 BACE1 (0.38) KMT2ABACE1CTSDALDH1A1
SCHEMBL7518290 0.81 LMNA (0.36) KMT2AP2RX7MEN1NPC1RAB9A
SCHEMBL7510378 0.79 ALDH1A1 (0.40) KMT2ABACE1CTSDMEN1RAB9A
SCHEMBL10144298 0.79 BACE1 (0.33) BACE1CTSD
SCHEMBL17551756 0.78 KMT2A (0.34) KMT2ABACE1CTSDMEN1ALDH1A1
SCHEMBL12504790 0.76 BACE1 (0.35) KMT2ABACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178513-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-15 US disclosed