SCHEMBL1014491

SCHEMBL1014491

CON(C)C(=O)c1ccc(CN2CCOCC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 3/20 0.61
EPAS1 Q99814 3/20 0.61
KMT2A Q03164 1/20 0.58
SMN1; SMN2 Q16637 3/20 0.56
MAPK1 P28482 1/20 0.56
HRH3 Q9Y5N1 2/20 0.55
TSHR P16473 1/20 0.55
HPGD P15428 1/20 0.54
KDM4E B2RXH2 1/20 0.53
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
LMNA P02545 1/20 0.51
TP53 P04637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1014092 0.85 ABL1 (0.50) HIF1AEPAS1KMT2ASMN1; SMN2HPGD
SCHEMBL1011847 0.84 MCHR1 (0.48) HIF1AEPAS1KMT2ASMN1; SMN2MAPK1
SCHEMBL25062318 0.82 HTT (0.63) HIF1AEPAS1KMT2ASMN1; SMN2MAPK1
SCHEMBL1421404 0.81 CTSB (0.50) HIF1AEPAS1KMT2ASMN1; SMN2MAPK1
SCHEMBL1014280 0.81 CYP2A13 (0.47) HIF1AEPAS1KMT2ASMN1; SMN2MAPK1
SCHEMBL1014530 0.80 MAPT (0.51) KMT2ASMN1; SMN2MAPK1KDM4ELMNA
SCHEMBL13674546 0.80 LTA4H (0.46) HIF1AEPAS1KMT2ASMN1; SMN2MAPK1
SCHEMBL1014528 0.80 HTT (0.54) KMT2ASMN1; SMN2LMNA
SCHEMBL171628 0.80 SMN1; SMN2 (0.81) HIF1AEPAS1KMT2ASMN1; SMN2MAPK1
SCHEMBL25062364 0.80 GSK3B (0.51) HIF1AKMT2ASMN1; SMN2MAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110034466-A1 NOVEL FIVE-MEMBERED RING COMPOUND DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-02-10 US disclosed
EP-2272835-A1 NOVEL FIVE-MEMBERED RING COMPOUND Dainippon Sumitomo Pharma Co., Ltd. (JP) 2011-01-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110034466-A1 NOVEL FIVE-MEMBERED RING COMPOUND CCL11, CCR1, CCR10 HIF1A 4335/4885EPAS1 2986/4885KMT2A 4321/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.