SCHEMBL10146347

SCHEMBL10146347

C=NC(=N)N1CCC(n2c(=O)n(C)c3cc(-c4ccccc4C)ccc32)CC1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.46
CTSS P25774 13/20 0.40
DRD2 P14416 1/20 0.40
SLC6A4 P31645 1/20 0.40
CYP3A4 P08684 1/20 0.38
TNKS O95271 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
PIK3CA P42336 1/20 0.37
MTOR P42345 1/20 0.37
PRKDC P78527 1/20 0.37
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20496328 0.86 HSD11B1 (0.51) HSD11B1CTSSDRD2SLC6A4CYP3A4
SCHEMBL14992429 0.83 HSD11B1 (0.53) HSD11B1DRD2SLC6A4CYP3A4TNKS
SCHEMBL10145862 0.81 PIK3CA (0.51) HSD11B1PIK3CAMTORPRKDC
SCHEMBL10145870 0.79 HTR7 (0.43) HSD11B1CTSSDRD2SLC6A4CYP3A4
SCHEMBL14992973 0.78 PIK3CA (0.51) HSD11B1CTSSDRD2SLC6A4PIK3CA
SCHEMBL14992428 0.76 HSD11B1 (0.41) HSD11B1CTSSDRD2SLC6A4CYP3A4
SCHEMBL10145863 0.67 PARP2 (0.47) HSD11B1DRD2SLC6A4PARP2PIK3CA
SCHEMBL10145954 0.67 PIK3CA (0.47) HSD11B1CTSSDRD2SLC6A4CYP3A4
SCHEMBL30724611 0.66 EZH2 (0.48) HSD11B1DRD2SLC6A4PARP2PIK3CA
SCHEMBL30724606 0.65 DRD2 (0.44) HSD11B1CTSSDRD2SLC6A4PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed