SCHEMBL10147136

SCHEMBL10147136

O=C(O)c1ccc2c(c1)C(=O)OC21CCN(c2ccc(-c3nc4cc(Cl)ccc4[nH]3)cn2)CC1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 17/20 0.73
KCNH2 Q12809 8/20 0.73
CYP2C9 P11712 1/20 0.60
ADORA2A P29274 2/20 0.46
NPY5R Q15761 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10147228 0.89 DGAT1 (0.89) DGAT1KCNH2CYP2C9
SCHEMBL10146443 0.88 DGAT1 (0.87) DGAT1KCNH2CYP2C9NPY5R
SCHEMBL10146480 0.86 DGAT1 (0.77) DGAT1KCNH2CYP2C9ADORA2ANPY5R
SCHEMBL10146489 0.84 DGAT1 (0.88) DGAT1KCNH2CYP2C9ADORA2ANPY5R
SCHEMBL10146550 0.82 DGAT1 (0.69) DGAT1KCNH2CYP2C9ADORA2ANPY5R
SCHEMBL10146482 0.82 DGAT1 (0.88) DGAT1KCNH2CYP2C9ADORA2ANPY5R
SCHEMBL4560992 0.81 DGAT1 (0.57) DGAT1KCNH2CYP2C9ADORA2A
SCHEMBL6993769 0.79 CHEK2 (0.53) DGAT1KCNH2CYP2C9ADORA2A
SCHEMBL10147294 0.78 DGAT1 (0.53) DGAT1KCNH2CYP2C9ADORA2A
SCHEMBL10082141 0.76 DGAT1 (0.49) DGAT1KCNH2CYP2C9ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009217-A1 SPIROCYCLIC COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed