SCHEMBL10147294

SCHEMBL10147294

O=C(O)c1ccc(C2=NOC3(CCN(c4ccc(-c5nc6cc(Cl)ccc6[nH]5)cn4)CC3)C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.53
KCNH2 Q12809 15/20 0.53
ADORA2A P29274 2/20 0.47
CYP2C9 P11712 4/20 0.46
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10147125 0.88 DGAT1 (0.58) DGAT1KCNH2CYP2C9CYP3A4
SCHEMBL4560992 0.83 DGAT1 (0.57) DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL10147136 0.78 DGAT1 (0.73) DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL14235553 0.78 DGAT1 (0.61) DGAT1KCNH2ADORA2A
SCHEMBL10146407 0.77 DGAT1 (0.72) DGAT1KCNH2ADORA2ACYP2C9CYP3A4
SCHEMBL4560928 0.77 DGAT1 (0.54) DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL6993769 0.76 CHEK2 (0.53) DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL10380674 0.76 DGAT1 (0.71) DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL1687858 0.76 DGAT1 (0.51) DGAT1KCNH2ADORA2ACYP3A4
SCHEMBL14235043 0.76 DGAT1 (0.59) DGAT1KCNH2ADORA2ACYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009217-A1 SPIROCYCLIC COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed