SCHEMBL6993769

SCHEMBL6993769

O=C(O)c1cccc(N2CCN(c3ccc(-c4nc5cc(Cl)ccc5[nH]4)cn3)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 4/20 0.53
DGAT1 O75907 12/20 0.52
KCNH2 Q12809 8/20 0.52
ADORA2A P29274 2/20 0.52
CYP2C9 P11712 1/20 0.46
MGLL Q99685 2/20 0.45
DRD2 P14416 1/20 0.45
DRD3 P35462 1/20 0.45
AURKA O14965 1/20 0.45
KDR P35968 1/20 0.45
AURKB Q96GD4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994359 0.90 CHEK2 (0.50) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL4560992 0.89 DGAT1 (0.57) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL10082141 0.88 DGAT1 (0.49) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL6994712 0.88 DGAT1 (0.54) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL14235068 0.85 DGAT1 (0.58) DGAT1KCNH2ADORA2A
SCHEMBL4543375 0.83 CHEK2 (0.59) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL14235558 0.83 DGAT1 (0.57) CHEK2DGAT1KCNH2ADORA2A
SCHEMBL10081925 0.82 MGLL (0.55) DGAT1KCNH2ADORA2ACYP2C9MGLL
SCHEMBL4543095 0.82 DGAT1 (0.53) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL4560928 0.82 DGAT1 (0.54) CHEK2DGAT1KCNH2ADORA2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed