SCHEMBL10148018

SCHEMBL10148018

COCCOCCC(=O)NC1CCC(N2C(=O)C=CC2=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.40
DRD2 P14416 12/20 0.38
DRD3 P35462 12/20 0.38
HTR2A P28223 9/20 0.38
HTR1A P08908 4/20 0.38
DRD4 P21917 4/20 0.38
HTR2B P41595 4/20 0.38
HTR2C P28335 3/20 0.38
DRD1 P21728 1/20 0.38
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
NAMPT P43490 1/20 0.36
SMYD3 Q9H7B4 1/20 0.35
KDM5A P29375 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4761681 0.83 CNR2 (0.38) CNR1CNR2
SCHEMBL12094075 0.77 NPSR1 (0.42) MAPTDRD2DRD3HTR2AHTR1A
SCHEMBL12094076 0.77 RAB9A (0.48) MAPTNPC1RAB9A
SCHEMBL10148045 0.76 POLB (0.34) MAPTDRD2DRD3HTR2AHTR1A
SCHEMBL4761695 0.76 MEN1 (0.39) MAPTDRD2DRD3HTR2AHTR1A
SCHEMBL10132074 0.75 SMN1; SMN2 (0.52) MAPTCNR1CNR2SMYD3
SCHEMBL25030885 0.74 NPSR1 (0.40) MAPTDRD2DRD3HTR2AHTR1A
SCHEMBL26062862 0.74 NPSR1 (0.40) MAPTDRD2DRD3HTR2AHTR1A
SCHEMBL23135471 0.73 NPSR1 (0.53) MAPTDRD2DRD3HTR2AHTR1A
SCHEMBL25029638 0.72 MME (0.40) MAPTDRD2DRD3HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8227555-B2 Hydrolytically stable maleimide-terminated polymers NEKTAR THERAPEUTICS (US) 2012-07-24 US disclosed
US-8106131-B2 Hydrolytically stable maleimide-terminated polymers NEKTAR THERAPEUTICS (US) 2012-01-31 US disclosed
US-20090012241-A1 Hydrolytically stable maleimide-terminated polymers NEKTAR THERAPEUTICS AL, CORPORATION (US) 2009-01-08 US disclosed
US-7432331-B2 Hydrolytically stable maleimide-terminated polymers NEKTAR THERAPEUTICS AL, CORPORATION (US) 2008-10-07 US disclosed
US-7432330-B2 Hydrolytically stable maleimide-terminated polymers NEKTAR THERAPEUTICS AL, CORPORATION (US) 2008-10-07 US disclosed