SCHEMBL10153642

SCHEMBL10153642

CCCNC(=O)C1C(=O)N(OCc2ccccc2)C(=O)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 2/20 0.42
FFAR1 O14842 1/20 0.40
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
TP53 P04637 1/20 0.38
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9958882 0.94 KMT2A (0.46) KCNA5FFAR1KMT2AMEN1MAPT
SCHEMBL10154063 0.93 KMT2A (0.47) KCNA5KMT2AMEN1MAPTALDH1A1
SCHEMBL9959019 0.92 KMT2A (0.47) KCNA5KMT2AMEN1MAPTALDH1A1
SCHEMBL10153579 0.92 KMT2A (0.47) KCNA5KMT2AMEN1MAPTALDH1A1
SCHEMBL9959738 0.92 KMT2A (0.47) KCNA5KMT2AMEN1MAPTALDH1A1
SCHEMBL9959313 0.88 KCNA5 (0.48) KCNA5KMT2AMEN1MAPTALDH1A1
SCHEMBL9959312 0.87 DRD2 (0.41) KCNA5KMT2AMEN1MAPTALDH1A1
SCHEMBL10153971 0.85 POLB (0.50) KCNA5KMT2AMEN1MAPTALDH1A1
SCHEMBL9959297 0.85 HDAC4 (0.49) KCNA5FFAR1KMT2AMEN1MAPT
SCHEMBL10153600 0.85 MAPT (0.44) KMT2AMEN1MAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed