SCHEMBL10167504

SCHEMBL10167504

COc1cccc2snc(N(C)C(=O)c3ccccc3)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.45
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
LMNA P02545 3/20 0.43
TP53 P04637 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
RAD52 P43351 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
KDM4E B2RXH2 2/20 0.40
OXTR P30559 1/20 0.39
PDE4D Q08499 1/20 0.37
HPGD P15428 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10167491 0.86 LMNA (0.40) NPC1RAB9ALMNATP53SMN1; SMN2
SCHEMBL10167509 0.84 RAD52 (0.51) KCNA5NPC1RAB9ATP53SMN1; SMN2
SCHEMBL10167444 0.84 KCNA5 (0.40) KCNA5NPC1RAB9ALMNATP53
SCHEMBL10167464 0.82 LMNA (0.45) NPC1RAB9ALMNATP53SMN1; SMN2
SCHEMBL10167501 0.81 KCNA5 (0.40) KCNA5NPC1RAB9ALMNASMN1; SMN2
SCHEMBL10167507 0.79 KDM4E (0.40) KCNA5NPC1RAB9ALMNATP53
SCHEMBL10167512 0.79 MAPT (0.39) KCNA5RAB9ATP53KDM4EHSD17B2
SCHEMBL13903746 0.78 KCNA5 (0.45) KCNA5NPC1RAB9ALMNATP53
SCHEMBL10167648 0.76 MAPT (0.59) KMT2AMEN1
SCHEMBL13903768 0.73 KCNA5 (0.44) KCNA5NPC1RAB9ATP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119568-B2 3-amino-1,2-benzisothiazole compounds for combating animal pest II BASF SE (DE) 2012-02-21 US disclosed
US-8119568-B2 3-amino-1,2-benzisothiazole compounds for combating animal pest II BASF SE (DE) 2012-02-21 US disclosed
US-20100009848-A1 3-Amino-1,2-Benzisothiazole Compounds for Combating Animal Pest II BASF SE (DE) 2010-01-14 US disclosed
US-20100009848-A1 3-Amino-1,2-Benzisothiazole Compounds for Combating Animal Pest II BASF SE (DE) 2010-01-14 US disclosed
WO-2008090048-A2 3-AMINO-1,2-BENZISOTHIAZOLE COMPOUNDS FOR COMBATING ANIMAL PEST II BASF SE (DE) 2008-07-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100009848-A1 3-Amino-1,2-Benzisothiazole Compounds for Combating Animal Pest II BPNT1, BCAT1, TGFBR1 KCNA5 1882/4885NPC1 2906/4885RAB9A 1949/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.