SCHEMBL1016771

SCHEMBL1016771

CS(=O)(=O)c1ccc(F)cc1CNC(=O)c1cc(Cl)c[nH]c1=N

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DDR1 Q08345 9/20 0.50
NTRK1 P04629 1/20 0.41
ADRA1D P25100 3/20 0.40
ADRA1A P35348 2/20 0.40
ADRA1B P35368 2/20 0.40
ROCK2 O75116 4/20 0.39
ROCK1 Q13464 4/20 0.39
CCR2 P41597 1/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RCE1 Q9Y256 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1017236 0.91 DDR1 (0.52) DDR1
SCHEMBL1018589 0.90 DDR1 (0.48) DDR1ADRA1D
Hydrochloric Acid SCHEMBL1018259 0.89 DDR1 (0.47) DDR1ADRA1D
SCHEMBL1017517 0.88 DDR1 (0.39) DDR1ADRA1DKDM4EALDH1A1RCE1
Hydrochloric Acid SCHEMBL1020060 0.88 DDR1 (0.39) DDR1ADRA1DKDM4EALDH1A1RCE1
Hydrochloric Acid SCHEMBL1018237 0.85 ALDH1A1 (0.45) ADRA1DKDM4EALDH1A1RCE1
Hydrochloric Acid SCHEMBL1017169 0.85 ALDH1A1 (0.46) ROCK2ROCK1KDM4EALDH1A1RCE1
Hydrochloric Acid SCHEMBL1017474 0.84 USP2 (0.46) DDR1ROCK2ROCK1ALDH1A1
SCHEMBL15703882 0.84 EPHX2 (0.46) DDR1ADRA1DROCK2ROCK1KDM4E
Hydrochloric Acid SCHEMBL1017391 0.84 EPHX2 (0.40) DDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271624-A1 IMINOPYRIDINE DERIVATIVES AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2011-01-12 EP disclosed
WO-2009131245-A1 IMINOPYRIDINE DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-29 WO disclosed