SCHEMBL10169109

SCHEMBL10169109

COc1cc(N)cc(C=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.48
NQO2 P16083 3/20 0.48
ALDH1A1 P00352 5/20 0.48
CYP2A6 P11509 1/20 0.48
CYP1A1 P04798 3/20 0.46
CYP1B1 Q16678 3/20 0.46
CYP3A4 P08684 1/20 0.42
ESR1 P03372 2/20 0.39
CYP1A2 P05177 2/20 0.39
TSHR P16473 1/20 0.39
ABL1 P00519 1/20 0.39
TTR P02766 1/20 0.39
ABCB1 P08183 1/20 0.39
ALOX5 P09917 1/20 0.39
BCR P11274 1/20 0.39
PTGS2 P35354 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
AHR P35869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL228003 0.84 CYP1A1 (0.64) CYP19A1NQO2ALDH1A1CYP2A6CYP1A1
SCHEMBL1663786 0.84 ALDH1A1 (0.58) CYP19A1NQO2ALDH1A1CYP2A6CYP1A1
Water SCHEMBL28227114 0.82 CYP1A1 (0.61) CYP19A1NQO2ALDH1A1CYP2A6CYP1A1
Formamide SCHEMBL28158838 0.80 ALDH1A1 (0.52) CYP19A1NQO2ALDH1A1CYP2A6CYP1A1
Formic Acid Methyl Ester SCHEMBL28071788 0.78 CYP1A1 (0.56) CYP19A1NQO2ALDH1A1CYP2A6CYP1A1
SCHEMBL378297 0.77 CYP1A1 (0.58) NQO2ALDH1A1CYP2A6CYP1A1CYP1B1
SCHEMBL29951799 0.77 ALDH1A1 (0.50) CYP19A1NQO2ALDH1A1CYP2A6CYP1A1
SCHEMBL5883049 0.77 ALDH1A1 (0.50) CYP19A1NQO2ALDH1A1CYP2A6CYP1A1
SCHEMBL29958196 0.77 CYP1A1 (0.58) NQO2ALDH1A1CYP2A6CYP1A1CYP1B1
SCHEMBL5800828 0.77 ALDH1A1 (0.59) CYP19A1NQO2ALDH1A1CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
CN-102952062-B Replace benzo-heterocycle compound and its preparation method and application 中国医学科学院医药生物技术研究所 2016-06-08 CN disclosed
CN-102952062-A Substituted benzoheterocyclic compounds and preparation method and application thereof INST MEDICINAL BIOTECHNOLOGY 2013-03-06 CN disclosed
WO-2012129423-A2 BIOMARKER DISCOVERY IN COMPLEX BIOLOGICAL FLUID USING BEAD OR PARTICLE BASED LIBRARIES AND DIAGNOSTIC KITS AND THERAPEUTICS OPKO PHARMACEUTICALS, LLC (US) 2012-09-27 WO disclosed
EP-2468743-A1 Nitrogen-containing bicyclic compounds useful as antibacterial agents Toyama Chemical Co., Ltd. (JP) 2012-06-27 EP disclosed
US-20120021530-A1 HETEROGENEOUS FOLDAMERS CONTAINING alpha, beta, and/or gamma-AMINO ACIDS WISCONSIN ALUMNI RESEARCH FOUNDATION 2012-01-26 US disclosed
WO-2010141421-A1 IDENTIFICATION OF SMALL MOLECULES RECOGNIZED BY ANTIBODIES IN SUBJECTS WITH NEURODEGENERATIVE DISEASES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-12-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120021530-A1 HETEROGENEOUS FOLDAMERS CONTAINING alpha, beta, and/or gamma-AMINO ACIDS DNPEP, PRKCSH, YWHAZ CYP19A1 3778/4885NQO2 1932/4885ALDH1A1 3160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.