SCHEMBL1017427

SCHEMBL1017427

O=C(O)[C@H]1CC1c1ccncc1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
NAMPT P43490 2/20 0.57
LMNA P02545 1/20 0.57
GAA P10253 1/20 0.57
HTT P42858 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
FFAR1 O14842 6/20 0.54
HDAC4 P56524 1/20 0.46
MAPT P10636 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ROCK2 O75116 2/20 0.43
SLC9A1 P19634 1/20 0.42
GPR88 Q9GZN0 1/20 0.41
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40
ITK Q08881 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1019296 1.00 ALDH1A1 (0.57) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL1017425 1.00 ALDH1A1 (0.57) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL1019924 0.84 ALDH1A1 (0.53) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL12765360 0.84 ALDH1A1 (0.53) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL1018424 0.84 ALDH1A1 (0.53) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL15219834 0.82 ALDH1A1 (0.51) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL30927243 0.82 ALDH1A1 (0.51) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL4126470 0.81 FFAR1 (0.70) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL5217474 0.81 FFAR1 (0.70) ALDH1A1NAMPTLMNAGAAHTT
SCHEMBL2034678 0.81 FFAR1 (0.70) ALDH1A1NAMPTLMNAGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271646-A1 APOPTOSIS SIGNAL-REGULATING KINASE 1 INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2011-01-12 EP disclosed
WO-2009123986-A1 APOPTOSIS SIGNAL-REGULATING KINASE 1 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-08 WO disclosed