SCHEMBL10175359

SCHEMBL10175359

Cn1c(-c2ccncc2)nc2ccc(Cl)cc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
RAB9A P51151 4/20 0.52
MAPT P10636 1/20 0.52
NPC1 O15118 3/20 0.50
KDM4E B2RXH2 1/20 0.50
CYP1A2 P05177 1/20 0.50
GAA P10253 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KCNH2 Q12809 1/20 0.50
AOC3 Q16853 1/20 0.50
CASP3 P42574 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
CYP11B1 P15538 2/20 0.48
CYP11B2 P19099 2/20 0.48
ATM Q13315 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10248874 0.84 MEN1 (0.66) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL17896659 0.83 MEN1 (0.59) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL17896686 0.82 CYP11B2 (0.71) MEN1KMT2ARAB9ANPC1KDM4E
SCHEMBL26603181 0.81 MEN1 (0.62) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL10175360 0.81 RAB9A (0.49) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL10175358 0.80 PDE10A (0.65) MEN1KMT2ARAB9AMAPTKDM4E
SCHEMBL10175361 0.80 PDE2A (0.52) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL10249413 0.79 MEN1 (0.63) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL17896687 0.79 CYP11B1 (0.55) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL17896692 0.79 CYP11B1 (0.46) MEN1KMT2ARAB9AMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed