SCHEMBL10175360

SCHEMBL10175360

Cc1cncc(-c2nc3ccc(Cl)cc3n2C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
MAPT P10636 1/20 0.49
CYP11B1 P15538 3/20 0.48
CYP11B2 P19099 2/20 0.48
NPC1 O15118 3/20 0.47
CASP3 P42574 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 2/20 0.43
CYP1A2 P05177 2/20 0.43
GAA P10253 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PTPN1 P18031 1/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896692 0.86 CYP11B1 (0.46) RAB9AMEN1KMT2AMAPTCYP11B1
SCHEMBL17896687 0.86 CYP11B1 (0.55) RAB9AMEN1KMT2AMAPTCYP11B1
SCHEMBL460358 0.84 RAB9A (0.48) RAB9AMEN1KMT2AMAPTCYP11B1
SCHEMBL10176203 0.83 CYP11B2 (0.69) MEN1KMT2ACYP11B1CYP11B2
SCHEMBL17896689 0.83 CYP11B2 (0.44) RAB9AMEN1KMT2AMAPTCYP11B1
SCHEMBL17883786 0.83 CYP11B2 (0.46) RAB9AMEN1KMT2AMAPTCYP11B1
SCHEMBL747042 0.83 CYP11B1 (0.43) RAB9AMEN1KMT2AMAPTCYP11B1
SCHEMBL17896694 0.82 FGFR3 (0.49) RAB9AMEN1KMT2AMAPTCYP11B1
SCHEMBL17896686 0.82 CYP11B2 (0.71) RAB9AMEN1KMT2ACYP11B1CYP11B2
SCHEMBL10175359 0.81 MEN1 (0.62) RAB9AMEN1KMT2AMAPTCYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed