SCHEMBL10175468

SCHEMBL10175468

CS(=O)(=O)Nc1ccc2c(c1)nc(-c1cccnc1)n2CCO

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.46
MAPK10 P53779 1/20 0.45
MAPT P10636 2/20 0.44
CYP17A1 P05093 1/20 0.43
KDM4E B2RXH2 1/20 0.43
HTT P42858 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
CTPS1 P17812 1/20 0.43
FYN P06241 1/20 0.43
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
NAMPT P43490 1/20 0.41
ALOX5AP P20292 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
F2 P00734 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175617 0.89 CYP11B2 (0.55) METMAPK10MAPTCYP17A1KDM4E
SCHEMBL460529 0.85 NAMPT (0.53) METMAPK10CYP17A1FYNCYP11B1
SCHEMBL10175462 0.85 KDM4E (0.42) KDM4EHTTHDAC1HDAC8CYP11B1
SCHEMBL17897056 0.84 MET (0.49) METMAPK10MAPTCYP17A1HTT
SCHEMBL17883790 0.80 USP2 (0.63) METMAPK10MAPTCYP17A1KDM4E
SCHEMBL10175612 0.78 CYP11B2 (0.63) METMAPK10CYP17A1CYP11B1CYP11B2
SCHEMBL17896765 0.74 CYP11B2 (0.58) MAPTKDM4EHTTCYP11B1CYP11B2
SCHEMBL17883783 0.73 CYP11B2 (0.43) MAPTKDM4EHTTCYP11B1CYP11B2
SCHEMBL10175134 0.73 CYP11B1 (0.59) HTTCYP11B1CYP11B2SMN1; SMN2CYP1A2
SCHEMBL14314688 0.72 CYP11B2 (0.56) MAPTKDM4ECYP11B1CYP11B2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed