SCHEMBL10175462

SCHEMBL10175462

CS(=O)(=O)Nc1ccc2c(c1)nc(-c1cncc(F)c1)n2CCO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
HTT P42858 1/20 0.42
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
DYRK1A Q13627 1/20 0.39
LMNA P02545 1/20 0.38
SIRT2 Q8IXJ6 3/20 0.38
SIRT1 Q96EB6 3/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 2/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
JAK3 P52333 1/20 0.37
PTGER4 P35408 1/20 0.37
BRPF1 P55201 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17883783 0.89 CYP11B2 (0.43) KDM4EHTTCNR1CNR2SMN1; SMN2
SCHEMBL17896755 0.85 SMN1; SMN2 (0.44) SMN1; SMN2DYRK1ALMNAALDH1A1POLB
SCHEMBL10175468 0.85 MET (0.46) KDM4EHTTCNR1CNR2SMN1; SMN2
SCHEMBL10175616 0.81 CYP11B1 (0.43) KDM4EHTTCNR1CNR2SMN1; SMN2
SCHEMBL459504 0.76 CYP11B2 (0.56) KDM4EHTTHDAC1HDAC8JAK2
SCHEMBL10175614 0.75 SMN1; SMN2 (0.46) SMN1; SMN2HDAC1HDAC8DYRK1ALMNA
SCHEMBL10175617 0.73 CYP11B2 (0.55) KDM4EHTTCNR1CNR2ALDH1A1
SCHEMBL17896651 0.72 CYP11B2 (0.48) KDM4EHTTSMN1; SMN2LMNAPTGER4
SCHEMBL17896756 0.71 PTGS2 (0.45) KDM4ESMN1; SMN2HDAC1HDAC8LMNA
SCHEMBL460529 0.69 NAMPT (0.53) SMN1; SMN2LMNAALDH1A1BRPF1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed