SCHEMBL10175583

SCHEMBL10175583

CCn1c(-c2cccnc2)nc2ccc(F)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 14/20 1.00
CYP11B1 P15538 13/20 1.00
RPS6KA5 O75582 1/20 0.52
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
NLRP3 Q96P20 1/20 0.45
BRD4 O60885 1/20 0.43
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175594 0.90 CYP11B2 (0.81) CYP11B2CYP11B1RPS6KA5CYP1A2CYP2C19
SCHEMBL17896586 0.87 CYP11B2 (0.77) CYP11B2CYP11B1CYP1A2CYP2C19TDP1
SCHEMBL17896590 0.86 CYP11B2 (0.75) CYP11B2CYP11B1CYP1A2CYP2C19TDP1
SCHEMBL10175584 0.85 CYP11B2 (1.00) CYP11B2CYP11B1
SCHEMBL10175585 0.83 CYP11B2 (0.71) CYP11B2CYP11B1
SCHEMBL10176164 0.83 CYP11B2 (1.00) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL12116699 0.82 CYP11B2 (0.70) CYP11B2CYP11B1RPS6KA5CYP1A2CYP2C19
SCHEMBL10175599 0.80 CYP11B2 (0.66) CYP11B2CYP11B1RPS6KA5
SCHEMBL10176165 0.80 CYP11B2 (1.00) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL20349192 0.77 CYP11B2 (1.00) CYP11B2CYP11B1RPS6KA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed