SCHEMBL10176165

SCHEMBL10176165

CC(C)n1c(-c2cccnc2)nc2ccc(F)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 17/20 1.00
CYP11B1 P15538 14/20 1.00
USP2 O75604 1/20 0.66
HTT P42858 1/20 0.66
NCOA1 Q15788 1/20 0.66
NCOA3 Q9Y6Q9 1/20 0.66
PDE10A Q9Y233 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896587 0.84 CYP11B2 (0.73) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10176164 0.83 CYP11B2 (1.00) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10175583 0.80 CYP11B2 (1.00) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10175587 0.79 CYP11B2 (1.00) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10176228 0.77 USP2 (0.70) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL460209 0.76 CYP11B2 (1.00) CYP11B2CYP11B1
SCHEMBL971842 0.76 PDE10A (0.67) CYP11B2CYP11B1PDE10A
SCHEMBL10175584 0.75 CYP11B2 (1.00) CYP11B2CYP11B1
SCHEMBL10176167 0.75 CYP11B2 (0.80) CYP11B2CYP11B1USP2HTTNCOA1
SCHEMBL10175131 0.74 USP2 (0.65) CYP11B2CYP11B1USP2HTTNCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed