SCHEMBL10177816

SCHEMBL10177816

Cc1ccc(-c2nc(C(F)(F)F)c[nH]2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
PTGS2 P35354 4/20 0.44
PTGS1 P23219 1/20 0.42
TDO2 P48775 1/20 0.41
HPGDS O60760 1/20 0.39
MAPK1 P28482 1/20 0.37
PDK2 Q15119 1/20 0.36
HDAC1 Q13547 3/20 0.35
HDAC6 Q9UBN7 3/20 0.35
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC8 Q9BY41 1/20 0.35
PSD A5PKW4 1/20 0.35
TLR7 Q9NYK1 1/20 0.34
TRPV4 Q9HBA0 1/20 0.34
PIK3CA P42336 2/20 0.33
PIK3CD O00329 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11623789 0.82 HPGD (0.43) NPC1RAB9ATRPV4
SCHEMBL25196918 0.82 CYP2A6 (0.38) TRPV4PIK3CAPIK3CDPIK3CBPI4KA
SCHEMBL30442899 0.82 DGAT1 (0.40) TRPV4PIK3CAPIK3CDPIK3CBPI4KA
SCHEMBL10177266 0.82 DGAT1 (0.40) TRPV4PIK3CAPIK3CDPIK3CBPI4KA
SCHEMBL27731893 0.81 NPBWR1 (0.44) PTGS2PTGS1
SCHEMBL22166069 0.81 TRPV4 (0.34) TRPV4PIK3CAPIK3CDPIK3CBPI4KA
SCHEMBL29429388 0.81 NPC1 (0.44) NPC1RAB9AMAPK1HDAC1HDAC6
SCHEMBL22165974 0.81 NPC1 (0.44) NPC1RAB9AMAPK1HDAC1HDAC6
SCHEMBL11621764 0.78 CCNC (0.40) PDK2
SCHEMBL11625195 0.77 NPY5R (0.47) NPC1RAB9APTGS2TDO2HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012081736-A1 CONTINUOUS ARYCYCLIC COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-06-21 WO disclosed
US-4125530-A FROM 1,1-DIHALO-3,3,3-TRIFLUOROACETONE, BASE, AMMONIA AND A CARBOXALDEHYDE MERCK & CO., INC. (US) 1978-11-14 US disclosed
US-4032522-A ANTI-GOUT, ANTI-HYPERURICEMIC MERCK & CO., INC. (US) 1977-06-28 US disclosed