SCHEMBL10179472

SCHEMBL10179472

Cc1ccc(F)c(-c2cccc(-c3ccnc(-c4ccc[nH]4)c3)c2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.61
TGFBR1 P36897 7/20 0.41
KDM4C Q9H3R0 1/20 0.40
MAPT P10636 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NPSR1 Q6W5P4 3/20 0.37
ALOX15 P16050 2/20 0.37
HPGD P15428 2/20 0.37
HSP90AA1 P07900 1/20 0.37
PIM1 P11309 1/20 0.37
NISCH Q9Y2I1 1/20 0.36
CASP3 P42574 2/20 0.36
SENP8 Q96LD8 2/20 0.36
SENP7 Q9BQF6 2/20 0.36
SENP6 Q9GZR1 2/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
NFKB1 P19838 1/20 0.36
CASP1 P29466 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17629076 0.82 KDR (0.52) KDRTGFBR1KDM4CMAPTSMN1; SMN2
SCHEMBL1460368 0.76 KDR (1.00) KDR
SCHEMBL11983623 0.74 CCR1 (0.57) KDRKDM4CPIM1MEN1KMT2A
SCHEMBL1461475 0.73 KDR (1.00) KDR
SCHEMBL20748504 0.72 KDM4C (0.49) KDRKDM4CMAPTHPGDMEN1
SCHEMBL20748703 0.72 KDR (0.56) KDRKDM4CMAPTALOX15MAPKAPK2
SCHEMBL13829512 0.69 ACHE (0.46) KDRSMN1; SMN2HPGDPIM1NISCH
SCHEMBL1460341 0.68 KDM4C (0.50) KDRKDM4CMAPKAPK2
SCHEMBL12203789 0.68 CYP3A4 (0.45) MAPTSMN1; SMN2NPSR1ALOX15HPGD
SCHEMBL4864306 0.67 MAPKAPK2 (0.41) KDRTGFBR1KDM4CPIM1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473501-A1 COMPOUNDS AS TYROSINE KINASE MODULATORS Allergan, Inc. (US) 2012-07-11 EP disclosed