SCHEMBL10183093

SCHEMBL10183093

CCn1c(C(C)(C)C)cnc1C

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.33
HSD17B10 Q99714 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
LMNA P02545 2/20 0.32
MAPK1 P28482 3/20 0.32
THRB P10828 1/20 0.32
TSHR P16473 1/20 0.32
RAD52 P43351 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
CCND2 P30279 1/20 0.30
CCND3 P30281 1/20 0.30
ALOX15 P16050 1/20 0.30
CASP1 P29466 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19497079 0.84 ALDH1A1 (0.33) KDM4ESMN1; SMN2ALDH1A1HPGDLMNA
SCHEMBL10183000 0.78 CYP1A2 (0.38) KDM4EALDH1A1HTTLMNARAD52
SCHEMBL10183096 0.78 CYP2C19 (0.31)
SCHEMBL10183100 0.76 HPGD (0.41) KDM4EHSD17B10SMN1; SMN2ALDH1A1HPGD
SCHEMBL14756121 0.73
SCHEMBL21936667 0.72
SCHEMBL10182976 0.71 RORC (0.33)
SCHEMBL10235421 0.70 MAPK1 (0.33) KDM4EHSD17B10SMN1; SMN2ALDH1A1LMNA
SCHEMBL12852029 0.69 KDM4E (0.34) KDM4EHSD17B10ALDH1A1HPGDCDK4
SCHEMBL24448757 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357208-A1 MYST FAMILY HISTONE ACETYLTRANSFERASE INHIBITORS Epizyme, Inc. (US) 2023-11-09 US disclosed
US-20230357208-A1 MYST FAMILY HISTONE ACETYLTRANSFERASE INHIBITORS Epizyme, Inc. (US) 2023-11-09 US disclosed
US-11685732-B2 MYST family histone acetyltransferase inhibitors Epizyme, Inc. (US) 2023-06-27 US disclosed
US-11685732-B2 MYST family histone acetyltransferase inhibitors Epizyme, Inc. (US) 2023-06-27 US disclosed
US-20220162197-A1 MYST FAMILY HISTONE ACETYLTRANSFERASE INHIBITORS Epizyme, Inc. 2022-05-26 US disclosed
US-20120040951-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS SUNESIS PHARMACEUTICALS, INC. 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220162197-A1 MYST FAMILY HISTONE ACETYLTRANSFERASE INHIBITORS EP300, KAT2A, KAT6A KDM4E 167/4885HSD17B10 1572/4885SMN1; SMN2 3017/4885
US-20230357208-A1 MYST FAMILY HISTONE ACETYLTRANSFERASE INHIBITORS EP300, KAT2A, KAT6A KDM4E 167/4885HSD17B10 1572/4885SMN1; SMN2 3017/4885
US-20120040951-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS BRAF, RAF1, ARAF KDM4E 2722/4885HSD17B10 1308/4885SMN1; SMN2 4529/4885
US-11685732-B2 MYST family histone acetyltransferase inhibitors EP300, KAT2A, KAT6A KDM4E 167/4885HSD17B10 1572/4885SMN1; SMN2 3017/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.