SCHEMBL10187134

SCHEMBL10187134

CN(CC1CC1)c1ncc(F)c(N)n1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 2/20 0.39
ACACB O00763 5/20 0.39
PDE10A Q9Y233 1/20 0.34
PAK4 O96013 4/20 0.31
PAK1 Q13153 4/20 0.31
AURKA O14965 1/20 0.31
DAO P14920 1/20 0.31
PTPN11 Q06124 1/20 0.30
CHRM4 P08173 1/20 0.30
BRD4 O60885 1/20 0.30
MERTK Q12866 1/20 0.30
CSF1R P07333 1/20 0.30
CCNK O75909 1/20 0.30
CSNK1A1 P48729 1/20 0.30
CDK7 P50613 1/20 0.30
CDK9 P50750 1/20 0.30
CDK13 Q14004 1/20 0.30
CDK12 Q9NYV4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20000500 0.75 ALDH1A1 (0.40)
SCHEMBL10187348 0.73 ACACB (0.41) NPY5RACACBPDE10APAK4PAK1
SCHEMBL20772888 0.70 DAO (0.36) NPY5RACACBPDE10ADAOBRD4
SCHEMBL12888681 0.69 GRIN2B (0.47) NPY5RACACBPDE10APAK4PAK1
SCHEMBL30018737 0.67 ACACB (0.41) NPY5RACACBPDE10APAK4PAK1
SCHEMBL13530424 0.67 DCK (0.48)
SCHEMBL10187135 0.66 NUDT1 (0.42) DAOBRD4CSF1R
SCHEMBL13593630 0.64 BRD4 (0.43) NPY5RACACBDAOBRD4CSF1R
SCHEMBL2388378 0.63 BRD4 (0.51) NPY5RPAK4PAK1AURKABRD4
SCHEMBL2388381 0.63 BRD4 (0.51) NPY5RPAK4PAK1AURKABRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed