SCHEMBL10187777

SCHEMBL10187777

O=C(NO)c1ccn(-c2ccccn2)c1Oc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
TSHR P16473 3/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
REN P00797 1/20 0.39
MMP2 P08253 2/20 0.39
MMP13 P45452 2/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP12 P39900 1/20 0.39
MMP14 P50281 1/20 0.39
MMP16 P51512 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAPK14 Q16539 1/20 0.38
MAPK8 P45983 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6531023 0.87 KMT2A (0.43) ALDH1A1KMT2AMEN1TSHRGAA
SCHEMBL16703428 0.85 CTNNB1 (0.43) ALDH1A1KMT2AMEN1TSHRGAA
SCHEMBL10187775 0.68 HDAC6 (0.44) HDAC8TDP1KDM4E
SCHEMBL6168541 0.64 NOTUM (0.45) ALDH1A1TSHRGAAPOLBKDM4E
SCHEMBL974435 0.64 CA12 (0.57) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL25060908 0.64 HDAC8 (0.57) KMT2AMEN1GAAMMP2MMP13
SCHEMBL974852 0.64 CTNNB1 (0.62) ALDH1A1KMT2AMEN1TSHRGAA
SCHEMBL2611428 0.63 TSHR (0.45) KMT2AMEN1TSHRGAAHDAC8
SCHEMBL25778552 0.62 L3MBTL1 (0.51) ALDH1A1TSHRGAAPOLBTDP1
SCHEMBL25778550 0.62 KDM4E (0.66) ALDH1A1TSHRGAAPOLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2473501-A1 COMPOUNDS AS TYROSINE KINASE MODULATORS Allergan, Inc. (US) 2012-07-11 EP disclosed