SCHEMBL10188239

SCHEMBL10188239

CCCC(C)Oc1ccc(N)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 6/20 0.48
TSHR P16473 3/20 0.47
MCHR1 Q99705 1/20 0.43
MAPK1 P28482 2/20 0.41
ALDH1A1 P00352 5/20 0.40
CYP3A4 P08684 3/20 0.40
MAPT P10636 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TEAD4 Q15561 1/20 0.38
PKM P14618 1/20 0.38
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDE4D Q08499 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
SIGMAR1 Q99720 2/20 0.35
GPR88 Q9GZN0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6651666 0.87 LMNA (0.45) TDP1TSHRALDH1A1CYP3A4MAPT
SCHEMBL30713022 0.85 TDP1 (0.43) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL10621067 0.85 TDP1 (0.43) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL23584099 0.84 TDP1 (0.48) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL13657967 0.84 GPR88 (0.40) MCHR1NPC1RAB9ASMN1; SMN2SIGMAR1
SCHEMBL6371042 0.83 TDP1 (0.50) TDP1TSHRMCHR1MAPK1ALDH1A1
SCHEMBL746308 0.83 TDP1 (0.50) TDP1TSHRMCHR1MAPK1ALDH1A1
SCHEMBL11338351 0.82 TAAR1 (0.52) CYP1A2
SCHEMBL20367612 0.82 TDP1 (0.43) TDP1TSHRMAPK1ALDH1A1CYP3A4
SCHEMBL4948726 0.82 TDP1 (0.48) TDP1TSHRMAPK1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed