SCHEMBL10189574

SCHEMBL10189574

O=C(CC1CCC(c2ccc(-c3ccc(-c4nc5cc(Cl)ccc5[nH]4)cc3)cc2)CC1)N1CCOCC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 12/20 0.61
SOAT1 P35610 3/20 0.61
TLR9 Q9NR96 1/20 0.46
TLR8 Q9NR97 1/20 0.46
TLR7 Q9NYK1 1/20 0.46
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 2/20 0.42
ALDH1A1 P00352 2/20 0.42
TP53 P04637 2/20 0.42
HPGD P15428 2/20 0.42
RAB9A P51151 2/20 0.42
HSD17B10 Q99714 2/20 0.42
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ACHE P22303 1/20 0.42
KCNH2 Q12809 3/20 0.41
ADORA2A P29274 1/20 0.41
ENPP2 Q13822 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10189107 0.75 DGAT1 (0.86) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189566 0.75 DGAT1 (0.77) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189573 0.74 DGAT1 (0.55) DGAT1SOAT1KDM4ENPC1ALDH1A1
SCHEMBL1687855 0.73 DGAT1 (0.60) DGAT1SOAT1KDM4EALDH1A1HSD17B10
SCHEMBL13163415 0.71 DGAT1 (0.44) DGAT1SOAT1TLR9TLR8TLR7
SCHEMBL10189113 0.70 DGAT1 (0.64) DGAT1SOAT1
SCHEMBL902462 0.70 DGAT1 (0.73) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL14434976 0.69 GRM5 (0.55)
SCHEMBL10326022 0.69 CHEK2 (0.54) DGAT1SOAT1MAPTSMN1; SMN2ACHE
SCHEMBL10189571 0.69 DGAT1 (0.40) DGAT1SOAT1TLR9TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed