SCHEMBL10189571

SCHEMBL10189571

CN1CCN(C(=O)CC2CCC(c3ccc(-c4ccc(-c5nc6cc(S(C)(=O)=O)ccc6[nH]5)c(F)c4)cc3)CC2)CC1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.40
SOAT1 P35610 2/20 0.40
KDM1A O60341 3/20 0.40
MAOB P27338 3/20 0.40
MAOA P21397 2/20 0.40
TLR9 Q9NR96 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
FASN P49327 2/20 0.36
SCD O00767 2/20 0.36
FADS1 O60427 1/20 0.36
MCHR1 Q99705 1/20 0.35
SLC6A9 P48067 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10188929 0.88 DGAT1 (0.52) DGAT1SOAT1SCDFADS1KCNH2
SCHEMBL901694 0.81 DGAT1 (0.52) DGAT1SOAT1SCDFADS1KCNH2
SCHEMBL10189113 0.77 DGAT1 (0.64) DGAT1SOAT1SCD
SCHEMBL10189649 0.75 DGAT1 (0.52) DGAT1SOAT1SCD
SCHEMBL10381835 0.75 DGAT1 (0.59) DGAT1KCNH2
SCHEMBL10189555 0.74 SCD (0.54) SCDFADS1
SCHEMBL10189215 0.73 DGAT1 (0.49) DGAT1SOAT1SCD
SCHEMBL14695340 0.71 GPR119 (0.56)
SCHEMBL10189564 0.71 DGAT1 (0.47) DGAT1SOAT1KCNH2
SCHEMBL10189574 0.69 DGAT1 (0.61) DGAT1SOAT1TLR9TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed