SCHEMBL10192249

SCHEMBL10192249

CC(C)(C)C1CCCc2ccc(C#N)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.44
KDM1A O60341 2/20 0.40
DRD2 P14416 4/20 0.39
DRD3 P35462 4/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PNMT P11086 2/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
CYP11B2 P19099 1/20 0.36
CYP3A4 P08684 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24593614 0.81 DRD2 (0.45) LRRK2KDM1ADRD2DRD3ALDH1A1
SCHEMBL15577017 0.81 DRD2 (0.45) LRRK2KDM1ADRD2DRD3ALDH1A1
SCHEMBL20706314 0.78 LRRK2 (0.44) LRRK2KDM1ADRD2DRD3PNMT
SCHEMBL6141623 0.76 CYP11B1 (0.49) LRRK2KDM1ADRD2DRD3ALDH1A1
SCHEMBL2818458 0.76 PGR (0.48) LRRK2KDM1ADRD2DRD3ALDH1A1
SCHEMBL15945555 0.76 HTR2A (0.44) LMNAPNMTNOS3NOS1NOS2
SCHEMBL24916200 0.74 CHRNA7 (0.48) KDM1A
SCHEMBL24593570 0.74 DRD2 (0.50) LRRK2KDM1ADRD2DRD3PNMT
SCHEMBL16906757 0.74 DRD2 (0.50) LRRK2KDM1ADRD2DRD3PNMT
SCHEMBL22872288 0.72 LRRK2 (0.41) LRRK2KDM1ACYP11B2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8674095-B2 Compounds for treating neuropsychiatric conditions AFRAXIS HOLDINGS, INC. (US) 2014-03-18 US disclosed
US-20120046283-A1 COMPOUNDS FOR TREATING NEUROPSYCHIATRIC CONDITIONS AFRAXIS INC. (US) 2012-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046283-A1 COMPOUNDS FOR TREATING NEUROPSYCHIATRIC CONDITIONS PAK2, PAK5, PAK6 LRRK2 111/4885KDM1A 1212/4885DRD2 1446/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.