SCHEMBL10192308

SCHEMBL10192308

C[C@@H](c1ccc(S(C)(=O)=O)cc1F)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.40
PTGS2 P35354 6/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
PSEN1 P49768 2/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36
NCSTN Q92542 2/20 0.36
APH1A Q96BI3 2/20 0.36
PSENEN Q9NZ42 2/20 0.36
PDE2A O00408 2/20 0.36
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 2/20 0.36
G6PD P11413 1/20 0.34
IDE P14735 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10105627 0.82 PTGS2 (0.43) KIF11PTGS2SMN1; SMN2PSEN1PSEN2
SCHEMBL23312355 0.77 PTGS2 (0.39) KIF11PTGS2AKR1C3AKR1C2
SCHEMBL10192373 0.75 HRH4 (0.39) PTGS2SMN1; SMN2
SCHEMBL22624027 0.74 PDE2A (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL18367838 0.73 PDE2A (0.41) PDE2A
SCHEMBL18367835 0.73 PDE2A (0.41) PDE2A
SCHEMBL16509490 0.72 KIF11 (0.39) KIF11PTGS2SMN1; SMN2AKR1C3AKR1C2
SCHEMBL646030 0.72 PTGS2 (0.56) KIF11PTGS2
SCHEMBL30041432 0.72 PTGS2 (0.56) KIF11PTGS2
SCHEMBL18367829 0.72 APLNR (0.46) PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8674095-B2 Compounds for treating neuropsychiatric conditions AFRAXIS HOLDINGS, INC. (US) 2014-03-18 US disclosed
US-20120046283-A1 COMPOUNDS FOR TREATING NEUROPSYCHIATRIC CONDITIONS AFRAXIS INC. (US) 2012-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046283-A1 COMPOUNDS FOR TREATING NEUROPSYCHIATRIC CONDITIONS PAK2, PAK5, PAK6 KIF11 835/4885PTGS2 2694/4885SMN1; SMN2 1157/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.