SCHEMBL10194102

SCHEMBL10194102

CO/C(N)=N/C(C)c1cc(NC(=O)c2ccc(N)cn2)ccc1F

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
BACE1 P56817 17/20 0.42
GRM4 Q14833 1/20 0.40
CTSD P07339 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194904 0.87 SMN1; SMN2 (0.42) SMN1; SMN2NPC1RAB9ABACE1
SCHEMBL10193857 0.86 BACE1 (0.51) BACE1
SCHEMBL10193244 0.86 BACE1 (0.53) BACE1CTSD
SCHEMBL10193709 0.81 SMN1; SMN2 (0.42) SMN1; SMN2BACE1GRM4
SCHEMBL10193576 0.78 NPC1 (0.43) SMN1; SMN2NPC1RAB9ABACE1GRM4
SCHEMBL10195044 0.76 SMN1; SMN2 (0.45) SMN1; SMN2NPC1RAB9ABACE1
SCHEMBL10193575 0.76 BACE1 (0.51) BACE1
SCHEMBL10193209 0.76 BACE1 (0.53) BACE1
SCHEMBL10193565 0.74 ALDH1A1 (0.39) SMN1; SMN2BACE1GRM4
SCHEMBL10194892 0.74 AURKA (0.43) SMN1; SMN2NPC1RAB9AGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415756-A1 ISOTHIOUREA DERIVATIVES OR ISOUREA DERIVATIVES HAVING BACE1 INHIBITORY ACTIVITY Shionogi&Co., Ltd. (JP) 2012-02-08 EP disclosed