SCHEMBL10197402

SCHEMBL10197402

CCC1CCC(c2ccc(-c3ccc4c(C(=O)Nc5ccc(C)cc5F)ccnc4c3)cc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.58
SOAT1 P35610 1/20 0.58
SOAT2 O75908 1/20 0.46
PREP P48147 3/20 0.38
KDR P35968 3/20 0.38
AXL P30530 2/20 0.37
MERTK Q12866 2/20 0.37
ABCB1 P08183 1/20 0.36
FLT1 P17948 2/20 0.35
CNR1 P21554 2/20 0.35
CNR2 P34972 2/20 0.35
HRH1 P35367 1/20 0.35
MRGPRX1 Q96LB2 1/20 0.35
MAPK14 Q16539 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10197380 0.92 DGAT1 (0.59) DGAT1SOAT1SOAT2PREPKDR
SCHEMBL10197379 0.83 DGAT1 (0.65) DGAT1SOAT1SOAT2PREPCNR1
SCHEMBL10198038 0.83 DGAT1 (0.72) DGAT1SOAT1SOAT2
SCHEMBL409812 0.83 DGAT1 (0.72) DGAT1SOAT1SOAT2
SCHEMBL409813 0.83 DGAT1 (0.72) DGAT1SOAT1SOAT2
SCHEMBL10197337 0.82 DGAT1 (0.83) DGAT1SOAT1SOAT2PREPKDR
SCHEMBL10197360 0.81 DGAT1 (0.62) DGAT1SOAT1SOAT2PREPCNR1
SCHEMBL10197400 0.81 DGAT1 (0.62) DGAT1SOAT1SOAT2PREPCNR1
SCHEMBL10197359 0.81 DGAT1 (0.66) DGAT1SOAT1SOAT2PREPKDR
SCHEMBL13190530 0.81 DGAT1 (0.54) DGAT1SOAT1PREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120022057-A1 BICYCLIC COMPOUNDS AS INHIBITORS OF DIACYGLYCEROL ACYLTRANSFERASE SCHERING CORPORATION (US) 2012-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120022057-A1 BICYCLIC COMPOUNDS AS INHIBITORS OF DIACYGLYCEROL ACYLTRANSFERASE DGAT2, DGAT1, LCAT DGAT1 2/4885SOAT1 18/4885SOAT2 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.