SCHEMBL1019979

SCHEMBL1019979

Cn1cc(OC(=O)Nc2ccc(F)cc2-c2ccc(Cl)c(Cl)c2)c(C(F)F)n1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 20/20 0.51
CHRM2 P08172 8/20 0.48
CHRM1 P11229 8/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1078423 0.94 CHRM3 (0.50) CHRM3CHRM2CHRM1
SCHEMBL1019145 0.93 CHRM3 (0.43) CHRM3CHRM2CHRM1
SCHEMBL5179370 0.89 CHRM3 (0.48) CHRM3CHRM2CHRM1
SCHEMBL1037091 0.87 CHRM3 (0.42) CHRM3CHRM2CHRM1
SCHEMBL4836876 0.86 CHRM3 (0.39) CHRM3CHRM2CHRM1
SCHEMBL1039642 0.85 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL5093432 0.85 CHRM3 (0.53) CHRM3CHRM2CHRM1
SCHEMBL68043 0.85 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL29349968 0.85 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL29445383 0.85 CHRM3 (0.51) CHRM3CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 106 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233000-B1 Post-harvest treatment BAYER IP GMBH (DE) 2016-07-13 EP claimed
EP-1909579-B1 FUNGICIDAL MIXTURES BASED ON AZOLOPYRIMIDINYLAMINES BASF SE (DE) 2015-10-07 EP claimed
EP-2097412-A2 FUNGICIDAL N-HETEROARYL-CONDENSED PYRIDINE DERIVATIVES AND FUNGICIDAL COMPOSITIONS BASF SE (DE) 2009-09-09 EP claimed
WO-2009071419-A1 FUNGICIDAL MIXTURES BASF SE (DE) 2009-06-11 WO claimed
WO-2008046856-A2 FUNGICIDAL COMPOSITIONS BASF SE (DE) 2008-04-24 WO claimed
EP-1912503-A2 FUNGICIDAL MIXTURES CONTAINING SUBSTITUTED 1-METHYL PYRAZOL-4-YL CARBOXYLIC ACID ANILIDES BASF SE (DE) 2008-04-23 EP claimed
EP-1912496-A1 FUNGICIDAL MIXTURES COMPRISING CARBOXYLIC ACID-N-[2-(HALOGENALK(ENYL)OXY)PHENYL]AMIDES BASF SE (DE) 2008-04-23 EP claimed
WO-2008040820-A2 FUNGICIDAL N-HETEROARYL-CONDENSED PYRIDINE DERIVATIVES AND FUNGICIDAL COMPOSITIONS BASF SE (DE) 2008-04-10 WO claimed
EP-1903869-A2 FUNGICIDE MIXTURES BASED ON 1-METHYL-PYRAZOL-4-YL CARBOXYLIC ACID ANILIDES BASF SE (DE) 2008-04-02 EP claimed
WO-2007017449-A1 FUNGICIDAL MIXTURES COMPRISING CARBOXYLIC ACID-N-[2-(HALOGENALK(ENYL)OXY)PHENYL]AMIDES BASF SE (DE) 2007-02-15 WO claimed
WO-2007017416-A2 FUNGICIDAL MIXTURES CONTAINING SUBSTITUTED 1-METHYL PYRAZOL-4-YL CARBOXYLIC ACID ANILIDES BASF SE (DE) 2007-02-15 WO claimed
WO-2007006806-A2 FUNGICIDE MIXTURES BASED ON 1-METHYL-PYRAZOL-4-YL CARBOXYLIC ACID ANILIDES BASF AKTIENGESELLSCHAFT (DE) 2007-01-18 WO claimed
WO-2007003643-A1 FUNGICIDAL MIXTURES BASED ON 3,4-DISUBSTITUTED PYRAZOLECARBOXYLIC ACID BIPHENYLAMIDES BASF AKTIENGESELLSCHAFT (DE) 2007-01-11 WO claimed
EP-2094080-B1 UTILISATION OF BLOCK COPOLYMERS BASED ON VINYL LACTAMES AND VINYL ACETATE AS SOLUBILISERS BASF SE (DE) 2017-06-07 EP disclosed
EP-2381770-B1 GEL FORMULA WHICH CAN BE STORED SAFELY FOR A LONG PERIOD WITH AT LEAST TWO ESSENTIALLY UNMIXED HYDROGELS BASF SE (DE) 2016-03-30 EP disclosed
EP-2259675-B1 FUNGICIDAL COMPOSITIONS COMPRISING 3'-BROMINE-2,3,4,6'-TETRAMETHOXY-2'-6-DIMETHYLBENZOPHENONE BASF SE (DE) 2015-10-07 EP disclosed
WO-2007012601-A1 6-PHENYL-PYRAZOLOPYRIMIDINE-7-YLAMINE FUNGICIDES BASF AKTIENGESELLSCHAFT (DE) 2007-02-01 WO disclosed
WO-2007006723-A1 7-AMINO-6-TETRAZOLYL-1,2,4-TRIAZOLO[1,5-A]PYRIMIDINE COMPOUNDS AND THEIR USE FOR CONTROLLING PATHOGENIC FUNGI BASF AKTIENGESELLSCHAFT (DE) 2007-01-18 WO disclosed
WO-2007006722-A1 2-SUBSTITUTED 7-AMINO-6-HETEROARYL-1, 2, 4-TRIAZOLO [1, 5-A] PYRIMIDINE COMPOUNDS AND THE USE THEREOF FOR CONTROLLING PATHOGENIC FUNGI BASF AKTIENGESELLSCHAFT (DE) 2007-01-18 WO disclosed
WO-2007003643-A1 FUNGICIDAL MIXTURES BASED ON 3,4-DISUBSTITUTED PYRAZOLECARBOXYLIC ACID BIPHENYLAMIDES BASF AKTIENGESELLSCHAFT (DE) 2007-01-11 WO disclosed