SCHEMBL1019145

SCHEMBL1019145

Cn1cc(OC(=O)Nc2cc(F)ccc2-c2ccc(Cl)c(Cl)c2)c(C(F)F)n1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 18/20 0.43
CHRM2 P08172 4/20 0.42
CHRM1 P11229 4/20 0.42
ADRB2 P07550 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
APP P05067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1019979 0.93 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL5179370 0.89 CHRM3 (0.48) CHRM3CHRM2CHRM1
SCHEMBL1078423 0.86 CHRM3 (0.50) CHRM3CHRM2CHRM1
SCHEMBL3036773 0.85 CHRM3 (0.43) CHRM3CHRM2CHRM1
SCHEMBL304334 0.85 CHRM3 (0.42) CHRM3CHRM2CHRM1PSEN1PSEN2
SCHEMBL29437140 0.85 CHRM3 (0.42) CHRM3CHRM2CHRM1PSEN1PSEN2
SCHEMBL5622869 0.83 CHRM3 (0.43) CHRM3
SCHEMBL4836876 0.82 CHRM3 (0.39) CHRM3CHRM2CHRM1
SCHEMBL3784960 0.80 CHRM3 (0.48) CHRM3CHRM2CHRM1
SCHEMBL3747983 0.80 LMNA (0.42) CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 117 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1909579-B1 FUNGICIDAL MIXTURES BASED ON AZOLOPYRIMIDINYLAMINES BASF SE (DE) 2015-10-07 EP claimed
EP-2348833-A2 LIQUID AQUEOUS CROP PROTECTION FORMULATIONS BASF SE (DE) 2011-08-03 EP claimed
WO-2010040834-A2 LIQUID AQUEOUS CROP PROTECTION FORMULATIONS BASF SE (DE) 2010-04-15 WO claimed
EP-2097412-A2 FUNGICIDAL N-HETEROARYL-CONDENSED PYRIDINE DERIVATIVES AND FUNGICIDAL COMPOSITIONS BASF SE (DE) 2009-09-09 EP claimed
WO-2008046856-A2 FUNGICIDAL COMPOSITIONS BASF SE (DE) 2008-04-24 WO claimed
EP-1909579-A1 FUNGICIDAL MIXTURES BASED ON AZOLOPYRIMIDINYLAMINES BASF SE (DE) 2008-04-16 EP claimed
WO-2008040820-A2 FUNGICIDAL N-HETEROARYL-CONDENSED PYRIDINE DERIVATIVES AND FUNGICIDAL COMPOSITIONS BASF SE (DE) 2008-04-10 WO claimed
EP-1903868-A1 FUNGICIDAL MIXTURES MADE FROM 1-METHYLPYRAZOL-4-YLCARBOXANILIDES BASF SE (DE) 2008-04-02 EP claimed
EP-1903867-A1 FUNGICIDE MIXTURES BASED ON 3,5-DISUBSTITUTED PYRAZOL-CARBOXYLIC ACID BIPHENYLAMIDES BASF SE (DE) 2008-04-02 EP claimed
EP-1901609-A2 FUNGICIDE MIXTURES BASED ON 3-MONOSUBSTITUTED PYRAZOLE CARBOXYLIC ACID BIPHENYL AMIDES BASF SE (DE) 2008-03-26 EP claimed
EP-1898703-A1 FUNGICIDE MIXTURES BASED ON 2,4-DISUBSTITUTED PYRAZOLE CARBOXYLIC ACID BIPHENYLAMIDES BASF SE (DE) 2008-03-19 EP claimed
EP-1819223-B1 USE OF MENADIONE FOR BOOSTING THE EFFECTIVENESS OF AGROCHEMICALS BASF SE (DE) 2008-03-12 EP claimed
EP-1813152-A1 Fungicidal mixture based on 3,4-disubstituted biphenylanilides BASF AKTIENGESELLSCHAFT (DE) 2007-08-01 EP claimed
EP-1813151-A1 Fungicidal compositions based on 1-methyl-pyrazol-4-yl-anilides BASF Aktiengesellschaft (DE) 2007-08-01 EP claimed
WO-2007012598-A1 FUNGICIDAL MIXTURES BASED ON AZOLOPYRIMIDINYLAMINES BASF AKTIENGESELLSCHAFT (DE) 2007-02-01 WO claimed
WO-2007003644-A1 FUNGICIDAL MIXTURES MADE FROM 1-METHYLPYRAZOL-4-YLCARBOXANILIDES BASF AKTIENGESELLSCHAFT (DE) 2007-01-11 WO claimed
WO-2007003603-A2 FUNGICIDE MIXTURES BASED ON 3-MONOSUBSTITUTED PYRAZOLE CARBOXYLIC ACID BIPHENYL AMIDES BASF AKTIENGESELLSCHAFT (DE) 2007-01-11 WO claimed
WO-2007003540-A1 FUNGICIDAL MIXTURES BASED ON 2,5-DISUBSTITUTED PYRAZOL CARBOXYLIC ACID BIPHENYLAMIDES BASF AKTIENGESELLSCHAFT (DE) 2007-01-11 WO claimed
WO-2007003564-A1 FUNGICIDE MIXTURES BASED ON 3,5-DISUBSTITUTED PYRAZOL-CARBOXYLIC ACID BIPHENYLAMIDES BASF AKTIENGESELLSCHAFT (DE) 2007-01-11 WO claimed
WO-2007000462-A1 FUNGICIDE MIXTURES BASED ON 2,4-DISUBSTITUTED PYRAZOLE CARBOXYLIC ACID BIPHENYLAMIDES BASF AKTIENGESELLSCHAFT (DE) 2007-01-04 WO claimed