SCHEMBL1078423

SCHEMBL1078423

Cn1cc(OC(=O)Nc2ccc(F)cc2-c2ccc(Cl)c(F)c2)c(C(F)F)n1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 20/20 0.50
CHRM2 P08172 9/20 0.42
CHRM1 P11229 9/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1019979 0.94 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL1037091 0.90 CHRM3 (0.42) CHRM3CHRM2CHRM1
SCHEMBL5622869 0.90 CHRM3 (0.43) CHRM3
SCHEMBL1019145 0.86 CHRM3 (0.43) CHRM3CHRM2CHRM1
SCHEMBL1077648 0.85 CHRM3 (0.50) CHRM3CHRM2CHRM1
SCHEMBL4836876 0.85 CHRM3 (0.39) CHRM3CHRM2CHRM1
SCHEMBL303047 0.85 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL29688317 0.85 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL5179370 0.82 CHRM3 (0.48) CHRM3CHRM2CHRM1
SCHEMBL3800595 0.81 CHRM3 (0.40) CHRM3CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071419-A1 FUNGICIDAL MIXTURES BASF SE (DE) 2009-06-11 WO claimed
WO-2009071389-A1 FUNGICIDE MIXTURES BASF SE (DE) 2009-06-11 WO claimed
WO-2009071450-A1 FUNGICIDAL MIXTURE BASF SE (DE) 2009-06-11 WO claimed
EP-2094080-B1 UTILISATION OF BLOCK COPOLYMERS BASED ON VINYL LACTAMES AND VINYL ACETATE AS SOLUBILISERS BASF SE (DE) 2017-06-07 EP disclosed
EP-2381770-B1 GEL FORMULA WHICH CAN BE STORED SAFELY FOR A LONG PERIOD WITH AT LEAST TWO ESSENTIALLY UNMIXED HYDROGELS BASF SE (DE) 2016-03-30 EP disclosed
EP-2271697-B1 ALCOHOL ALKOXYLATES, MEDIA CONTAINING THESE AND UTILISATION OF ALCOHOL ALKOXYLATES AS ADJUVANTS FOR THE AGROCHEMICAL SECTOR BASF SE (DE) 2014-07-09 EP disclosed
EP-2046784-B1 AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME BASF SE (DE) 2011-09-14 EP disclosed
EP-2069413-B1 ACTIVE INGREDIENT FORMULATIONS CONTAINING COMB POLYMERS BASF SE (DE) 2011-08-03 EP disclosed
EP-2278877-A2 CYCLODEXTRIN-CONTAINING SUSPENSION CONCENTRATES, METHOD FOR PRODUCING THE SAME AND THEIR USE BASF SE (DE) 2011-02-02 EP disclosed
EP-2041125-B1 AZOLYLMETHYLOXIRANES, THEIR USE FOR CONTROLLING PHYTOPATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUNDS BASF SE (DE) 2011-01-26 EP disclosed
EP-2271697-A1 ALCOHOL ALKOXYLATES, AGENTS COMPRISING THE SAME AND USE OF THE ALCOHOL ALKOXYLATES AS ADJUVANTS IN THE AGROCHEMICAL FIELD BASF SE (DE) 2011-01-12 EP disclosed
WO-2008040786-A1 COMB POLYMERS AND USE THEREOF FOR THE PRODUCTION OF ACTIVE OR EFFECTIVE INGREDIENT FORMULATIONS BASF SE (DE) 2008-04-10 WO disclosed
WO-2008037607-A1 HETEROCYCLIC COMPOUNDS CONTAINING CARBONYL GROUPS, AND THE USE THEREOF FOR CONTROLLING PHYTOPATHOGENIC FUNGI BASF SE (DE) 2008-04-03 WO disclosed
WO-2008012246-A1 AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME BASF SE (DE) 2008-01-31 WO disclosed
WO-2008012234-A2 AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME BASF SE (DE) 2008-01-31 WO disclosed
WO-2008003607-A1 AZOLYLMETHYLOXIRANES, THEIR USE FOR CONTROLLING PHYTOPATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUNDS BASF SE (DE) 2008-01-10 WO disclosed
WO-2008003622-A1 AZOLYLMETHYLOXIRANES, THEIR USE FOR CONTROLLING PHYTOPATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUNDS BASF SE (DE) 2008-01-10 WO disclosed
WO-2007113136-A1 USE OF SUBSTITUTED TRIAZOLOPYRIMIDINES FOR CONTROLLING PHYTOPATHOGENIC HARMFUL FUNGI BASF AKTIENGESELLSCHAFT (DE) 2007-10-11 WO disclosed
WO-2007101804-A1 SUBSTITUTED PYRAZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF AND USE THEREOF FOR CONTROLLING PARASITIC FUNGI AND AGENTS COMPRISING THE SAME BASF SE (DE) 2007-09-13 WO disclosed
WO-2007101810-A1 SUBSTITUTED TRIAZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF AND USE THEREOF FOR CONTROLLING PARASITIC FUNGI AND AGENTS CONTAINING THE SAME BASF SE (DE) 2007-09-13 WO disclosed