SCHEMBL1019992

SCHEMBL1019992

N#CCc1cc(F)cc(F)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
IDO1 P14902 2/20 0.41
ENPP2 Q13822 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
MMP3 P08254 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
DAO P14920 2/20 0.32
CSNK2A1 P68400 1/20 0.31
DBH P09172 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8657492 0.95 KDM4E (0.43) KDM4ETDP1IDO1ENPP2CYP11B1
SCHEMBL14431663 0.86 KDM4E (0.38) KDM4ETDP1IDO1ENPP2CYP11B1
SCHEMBL1469433 0.85 TAAR1 (0.46) KDM4ETDP1IDO1CYP11B1CYP11B2
SCHEMBL332715 0.84 KDM4E (0.37) KDM4ETDP1IDO1ENPP2CYP11B1
SCHEMBL1072135 0.84 KDM4E (0.41) KDM4ETDP1IDO1ENPP2CYP11B1
SCHEMBL25170271 0.84 CA12 (0.48) KDM4ETDP1IDO1ENPP2CYP11B1
SCHEMBL25808872 0.84 KDM4E (0.37) KDM4ETDP1IDO1ENPP2CYP11B1
SCHEMBL1401399 0.84 CYP4F2 (0.41) KDM4ETDP1IDO1ENPP2CYP11B1
SCHEMBL20576683 0.84 KDM4E (0.37) KDM4ETDP1IDO1ENPP2CYP11B1
SCHEMBL25990556 0.84 KDM4E (0.37) KDM4ETDP1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 216 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12577245-B2 Sulfonyl benzamide derivatives as Bcl-2 inhibitors ASCENTAGE PHARMA (SUZHOU) CO., LTD. (CN) 2026-03-17 US disclosed
CN-120184379-A Flame-retardant electrolyte and preparation method thereof 抚顺国腾润滑科技有限公司 2025-06-20 CN disclosed
WO-2025104443-A1 INHIBITORY COMPOUNDS STORM THERAPEUTICS LTD (GB) 2025-05-22 WO disclosed
CN-119874565-A Mono cyano diaryl ethylene preparation method of class compound 常州大学 2025-04-25 CN disclosed
US-20250122171-A1 Substituted Amine Compounds, Compositions and Methods of Use DEEP APPLE THERAPEUTICS, INC. 2025-04-17 US disclosed
WO-2025064534-A1 SUBSTITUTED AMINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE DEEP APPLE THERAPEUTICS, INC. (US) 2025-03-27 WO disclosed
CN-116854668-B Phthalazinone compound, pharmaceutical composition and application thereof 中国药科大学 2025-02-07 CN disclosed
US-20240166644-A1 SULFONYL BENZAMIDE DERIVATIVES AS BCL-2 INHIBITORS ASCENTAGE PHARMA GROUP CORP LIMITED (CN) 2024-05-23 US disclosed
CN-115677731-B Organic compound and application thereof in organic electronic device 广州追光科技有限公司 2024-04-16 CN disclosed
US-20240004296-A1 RESIST UNDERLAYER FILM-FORMING COMPOSITION NISSAN CHEMICAL CORPORATION (JP) 2024-01-04 US disclosed
US-6506782-B1 Compounds which inhibit beta -amyloid peptide release and/or its synthesis, and, accordingly, have utility in treating Alzheimer's disease. Also disclosed are pharmaceutical compositions comprising a compound which inhibits beta ATHENA NEUROSCIENCES, INC. 2003-01-14 US disclosed
EP-0787127-B1 5-LIPOXYGENASE INHIBITORS PFIZER (US) 2001-01-03 EP disclosed
CN-1253554-A Heterocyclic compounds and their use for inhibiting 'beta'-amyloid peptide ELAN MEDICINE CO (US) 2000-05-17 CN disclosed
US-6063928-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS, CARDIOTONIC AGENTS PFIZER INC (US) 2000-05-16 US disclosed
EP-0968198-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR INHIBITING $g(b)-AMYLOID PEPTIDE Elan Pharmaceuticals, Inc. (US) 2000-01-05 EP disclosed
US-5883106-A 5-lipoxygenase inhibitors PFIZER INC. (US) 1999-03-16 US disclosed
WO-1998038177-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR INHIBITING β-AMYLOID PEPTIDE ELAN PHARMACEUTICALS, INC. (US) 1998-09-03 WO disclosed
EP-0787127-A1 5-LIPOXYGENASE INHIBITORS PFIZER INC. (US) 1997-08-06 EP disclosed
WO-1996011911-A1 5-LIPOXYGENASE INHIBITORS PFIZER INC. (US) 1996-04-25 WO disclosed
CN-1119099-A Method for preparing pharmacologically active CNS composition WELLCOME FOUND (GB) 1996-03-27 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12577245-B2 Sulfonyl benzamide derivatives as Bcl-2 inhibitors BCL2A1, BCL2L1, BCL2L11 KDM4E 3052/4885TDP1 3142/4885IDO1 4206/4885
US-20250122171-A1 Substituted Amine Compounds, Compositions and Methods of Use MRGPRX2, MRGPRX1, MRGPRX4 KDM4E 3489/4885TDP1 2286/4885IDO1 2668/4885
US-20240166644-A1 SULFONYL BENZAMIDE DERIVATIVES AS BCL-2 INHIBITORS BCL2, BCL2L2, BCL2L1 KDM4E 1780/4885TDP1 2368/4885IDO1 4546/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.