SCHEMBL1021565

SCHEMBL1021565

CS(=O)(=O)N1CCN(CC(O)CN2C3C[CH]C[C@@]2(C(N)=O)CC3)CC1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 16/20 0.37
HTR3A P46098 10/20 0.36
CYP2D6 P10635 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PRMT5 O14744 2/20 0.32
WDR77 Q9BQA1 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2980596 1.00 HTR4 (0.37) HTR4HTR3ACYP2D6SMN1; SMN2PRMT5
SCHEMBL1022503 1.00 HTR4 (0.37) HTR4HTR3ACYP2D6SMN1; SMN2PRMT5
SCHEMBL1022505 1.00 HTR4 (0.37) HTR4HTR3ACYP2D6SMN1; SMN2PRMT5
SCHEMBL3983379 0.90 HRH3 (0.32) HTR4
SCHEMBL3986065 0.90 HRH3 (0.32) HTR4
SCHEMBL3983380 0.88 KDM4E (0.38) CYP2D6SMN1; SMN2
SCHEMBL3986069 0.88 KDM4E (0.38) CYP2D6SMN1; SMN2
SCHEMBL3979933 0.88 CYP2D6 (0.32) CYP2D6SMN1; SMN2
SCHEMBL2980473 0.87 CYP2D6 (0.31) CYP2D6SMN1; SMN2
SCHEMBL2975908 0.85 PIK3CD (0.37) PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902053-B1 BENZOIMIDAZOLONE-CARBOXAMIDE COMPOUNDS AS 5-HT4 RECEPTOR AGONISTS THERAVANCE INC (US) 2011-01-12 EP claimed