SCHEMBL1022261

SCHEMBL1022261

S=C=Nc1ccccc1Br

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
CYP3A4 P08684 2/20 0.52
HPGD P15428 2/20 0.52
ABCB11 O95342 1/20 0.52
NR3C1 P04150 1/20 0.52
CYP1A2 P05177 1/20 0.52
ADRA2A P08913 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
ALOX15 P16050 1/20 0.52
ADRA2C P18825 1/20 0.52
MAOA P21397 1/20 0.52
DRD1 P21728 1/20 0.52
SLC6A4 P31645 1/20 0.52
HTR2B P41595 1/20 0.52
CCR2 P41597 1/20 0.52
HSD17B10 Q99714 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
MIF P14174 2/20 0.46
POLB P06746 2/20 0.43
APLNR P35414 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30507607 1.00 ALDH1A1 (0.52) ALDH1A1CYP3A4HPGDABCB11NR3C1
SCHEMBL207554 0.82 ALDH1A1 (0.62) ALDH1A1CYP3A4HPGDABCB11NR3C1
SCHEMBL29374052 0.82 ALDH1A1 (0.62) ALDH1A1CYP3A4HPGDABCB11NR3C1
SCHEMBL11436625 0.80 MEN1 (0.42) ALDH1A1CYP3A4HPGDABCB11NR3C1
SCHEMBL27995840 0.79 ALDH1A1 (0.46) ALDH1A1CYP3A4HPGDABCB11NR3C1
SCHEMBL29463737 0.76 CYP3A4 (0.52) ALDH1A1CYP3A4HPGDTDP1POLB
SCHEMBL6137454 0.76 MEN1 (0.36) ALDH1A1POLBMEN1KMT2ANPC1
SCHEMBL93220 0.76 CYP3A4 (0.52) ALDH1A1CYP3A4HPGDTDP1POLB
SCHEMBL4466979 0.75 ALDH1A1 (0.56) ALDH1A1CYP3A4HPGDABCB11NR3C1
SCHEMBL22588550 0.74 APLNR (0.47) ALDH1A1CYP3A4HPGDABCB11NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 243 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117924210-A Preparation method of 2-iminothiazolidine-4-ketone compound 赣南师范大学 2024-04-26 CN claimed
CN-117247409-A 3-thio/seleno-phosphorylated imidazole derivative and synthetic method and application thereof 曲阜师范大学 2023-12-19 CN claimed
CN-111471171-A Aryl sulfonic acid intermediate, preparation method thereof and application thereof in synthesizing low-temperature-sensitivity additive for concrete 江苏苏博特新材料股份有限公司 2020-07-31 CN claimed
CN-109265382-A A kind of fluorine-containing thiocarbamates compound and its synthetic method 湖北科技学院 2019-01-25 CN claimed
CN-107188866-A A kind of synthetic method of the ketone compounds of polysubstituted thiazole 4 湖北科技学院 2017-09-22 CN claimed
CN-106966990-A A kind of synthetic method of the polysubstituted ketone compounds of 2 thiocarbamoyl imidazole quinoline 4 湖北科技学院 2017-07-21 CN claimed
US-20160250175-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE JC (WUXI) COMPANY, INC. (CN) 2016-09-01 US claimed
EP-3034076-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE JC (Wuxi) COMPANY, Inc. (CN) 2016-06-22 EP claimed
CN-105267967-A Combined application of isothiocyanate-type compound and anti-cancer drug acting or affecting DNA WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2016-01-27 CN claimed
CN-104415332-A Combined application between isothiocyanate-type compound and kinase inhibitor medicine in treatment of cancer WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2015-03-18 CN claimed
CN-104117064-A Combined application of isothiocyanate compound and hormone medicine WUXI JC PHARMACAUTICAL TECHNOLOGY INC 2014-10-29 CN claimed
WO-2010065329-A2 NANOPARTICLES FOR CANCER TREATMENT THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-06-10 WO claimed
US-20060241178-A1 Compositions and methods for treating lung cancer IMMUNEGUARD LLC (US) 2006-10-26 US claimed
WO-2004060365-A1 COMPOSITIONS AND METHODS FOR TREATING LUNG CANCER AMERICAN HEALTH FOUNDATION (US) 2004-07-22 WO claimed
US-12515188-B2 Automated microreactor for effective optimization of high-speed chemical reaction, and method of optimizing high-speed chemical reaction therefor POSTECH Research and Business Development Foundation (KR) 2026-01-06 US disclosed
US-20250188046-A1 ULTRAFAST FLOW SYNTHESIS OF FUNCTIONALIZED SULFONYL FLUORIDES AND SUBSEQUENT SUFEX CONNECTIONS VIA LITHIATED CHEMISTRY POSTECH Research and Business Development Foundation (KR) 2025-06-12 US disclosed
EP-3446689-B1 ISOTHIOCYANATE COMPOUND FOR USE IN THE TREATMENT OF HYPERBILIRUBINEMIA JC WUXI COMPANY INC (CN) 2025-01-08 EP disclosed
EP-0416820-A2 Novel compounds exhibiting a vasodilating activity and inhibitory activity for platelet aggregation and pharmaceutical compositions containing them Hidaka, Hiroyoshi (JP) 1991-03-13 EP disclosed
EP-0352812-A1 Antiarthritic alpha-arylcarbamoyl cyanoacetic acid derivatives Bristol-Myers Squibb Company (US) 1990-01-31 EP disclosed
EP-0349243-A2 Antiviral combinations and compounds therefor THE WELLCOME FOUNDATION LIMITED (GB) 1990-01-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160250175-A1 COMBINED APPLICATION OF ISOTHIOCYANATE COMPOUND AND ANTI-CANCER MEDICINE CHUK, KIT, MKI67 ALDH1A1 2081/4885CYP3A4 2452/4885HPGD 3624/4885
US-20250188046-A1 ULTRAFAST FLOW SYNTHESIS OF FUNCTIONALIZED SULFONYL FLUORIDES AND SUBSEQUENT SUFEX CONNECTIONS VIA LITHIATED CHEMISTRY FGFR4, STS, FGFR1 ALDH1A1 1626/4885CYP3A4 644/4885HPGD 4811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.