SCHEMBL10229093

SCHEMBL10229093

Cc1[nH]c(=O)c2cc(Cl)ccc2c1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.58
LMNA P02545 2/20 0.47
TP53 P04637 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CYP1A2 P05177 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
CHEK1 O14757 2/20 0.44
TYMS P04818 3/20 0.43
DAO P14920 2/20 0.43
LCK P06239 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
PIM1 P11309 1/20 0.40
PIM2 Q9P1W9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1721110 0.77 ADRA2A (0.50) PARP1LMNATP53SMN1; SMN2CYP1A2
SCHEMBL10229086 0.76 PARP1 (0.44) PARP1LMNATP53SMN1; SMN2CYP1A2
SCHEMBL13901568 0.76 PARP1 (0.47) PARP1LMNATP53SMN1; SMN2CYP1A2
Iodide SCHEMBL1720068 0.75 PARP1 (0.46) PARP1LMNATP53SMN1; SMN2CYP1A2
SCHEMBL9843379 0.75 LMNA (0.56) LMNACYP1A2GAAHPGDCHEK1
SCHEMBL30547019 0.75 LMNA (0.56) LMNACYP1A2GAAHPGDCHEK1
SCHEMBL8288846 0.75 TP53 (0.56) PARP1LMNATP53SMN1; SMN2CYP1A2
SCHEMBL1720536 0.74 PARP1 (0.45) PARP1LMNATP53SMN1; SMN2CYP1A2
SCHEMBL9384092 0.73 PARP1 (1.00) PARP1LMNATP53SMN1; SMN2CYP1A2
SCHEMBL4078132 0.73 PARP1 (0.44) PARP1LMNATP53SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1566380-B1 ISOQUINOLINE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI TANABE PHARMA CORP (JP) 2012-01-11 EP disclosed