SCHEMBL9843379

SCHEMBL9843379

Cc1[nH]c2ccc(Cl)cc2c1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.56
HPGD P15428 2/20 0.55
CYP1A2 P05177 1/20 0.55
GAA P10253 1/20 0.55
HTR6 P50406 3/20 0.54
HTR7 P34969 2/20 0.54
ADRA2A P08913 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
HTR2B P41595 1/20 0.54
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
THRB P10828 1/20 0.53
SIRT1 Q96EB6 1/20 0.53
AHR P35869 1/20 0.52
MAPT P10636 2/20 0.51
IDO1 P14902 1/20 0.49
HTR1B P28222 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30547019 1.00 LMNA (0.56) LMNAHPGDCYP1A2GAAHTR6
SCHEMBL3632803 0.84 LMNA (0.53) LMNAHPGDCYP1A2GAAHTR6
Hydrochloric Acid SCHEMBL21724904 0.84 SIRT1 (0.45) LMNAHPGDCYP1A2GAAHTR6
SCHEMBL8288846 0.83 TP53 (0.56) LMNAHPGDCYP1A2GAAHTR6
SCHEMBL21980641 0.82 LMNA (0.55) LMNAHPGDCYP1A2GAAHTR6
SCHEMBL1757618 0.80 LMNA (0.53) LMNAHPGDCYP1A2GAAHTR6
SCHEMBL13997300 0.80 SIRT1 (0.54) LMNAHPGDCYP1A2GAAHTR6
SCHEMBL13174592 0.78 ALDH1A1 (0.56) LMNAHPGDGAAALDH1A1KDM4E
SCHEMBL30547023 0.78 ALDH1A1 (0.56) LMNAHPGDGAAALDH1A1KDM4E
SCHEMBL16688229 0.78 KDM4E (0.57) LMNAHPGDALDH1A1KDM4ETHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12371429-B2 Antibiotic resistance-modifying tricyclic heteroaryl compounds and uses thereof RECREO PHARMACEUTICALS LLC (US) 2025-07-29 US disclosed
CN-118344279-B Synthesis method of indole C2 benzyl C-H bond direct amine methylation 山东第二医科大学 2024-08-30 CN disclosed
CN-118344279-A Synthesis method of indole C2 benzyl C-H bond direct amine methylation 山东第二医科大学 2024-07-16 CN disclosed
CN-116730814-A Novel naphthoquinone intermediate, preparation method thereof, chiral naphthalene compound and preparation method thereof 香港科技大学深圳研究院 2023-09-12 CN disclosed
CN-110878099-B Preparation method of pyrrole [1,2, alpha ] indole alkaloid derivative 五邑大学 2021-11-30 CN disclosed
WO-2021145729-A1 NOVEL COMPOUND, PREPARATION METHOD THEREOF, AND USE THEREOF DAEGU-GYEONGBUK MEDICAL INNOVATION FOUNDATION (KR) 2021-07-22 WO disclosed
US-20210163479-A1 1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOLE DERIVATIVE COMPOUNDS AND USES THEREOF RECREO PHARMACEUTICALS LLC (US) 2021-06-03 US disclosed
US-20210163479-A1 1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOLE DERIVATIVE COMPOUNDS AND USES THEREOF RECREO PHARMACEUTICALS LLC (US) 2021-06-03 US disclosed
CN-112654354-A 1,3,4, 9-tetrahydro-2H-pyrido [3,4-b ] indole derivative compound and application thereof 菲尼克思药业股份有限公司 2021-04-13 CN disclosed
CN-110437126-B Organocatalytic indole non-activated sp3Method and application for asymmetric functionalization of carbon-hydrogen bond 香港科技大学深圳研究院 2020-11-13 CN disclosed
WO-2020037155-A1 1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOLE DERIVATIVE COMPOUNDS AND USES THEREOF RECREO PHARMACEUTICALS LLC (US) 2020-02-20 WO disclosed
CN-110437126-A Organic catalysis indoles disactivation sp3The method and application of C-H bond asymmetry function dough HKUST SHENZHEN RES INSTITUTE 2019-11-12 CN disclosed
US-8148392-B2 2-indolyl imidazo [4,5-d] phenanthroline derivatives and their use in the treatment of cancer LORUS THERAPEUTICS INC. (CA) 2012-04-03 US disclosed
US-8148392-B2 2-indolyl imidazo [4,5-d] phenanthroline derivatives and their use in the treatment of cancer LORUS THERAPEUTICS INC. (CA) 2012-04-03 US disclosed
WO-2010102393-A1 2-INDOLYL IMIDAZO [4,5-D]PHENANTHROLINE DERIVATIVES AND THEIR USE TO INHIBIT ANGIOGENESIS LORUS THERAPEUTICS INC. (CA) 2010-09-16 WO disclosed
US-20100168417-A1 2-Indolyl Imidazo [4,5-d] Phenanthroline Derivatives and Their Use in the Treatment for Cancer APTOSE BIOSCIENCES INC. (CA) 2010-07-01 US disclosed
US-20100168417-A1 2-Indolyl Imidazo [4,5-d] Phenanthroline Derivatives and Their Use in the Treatment for Cancer APTOSE BIOSCIENCES INC. (CA) 2010-07-01 US disclosed
EP-0425345-A1 Keratinic fibres dyeing process with amino-indoles, composition and use devices L'OREAL (FR) 1991-05-02 EP disclosed
US-4069337-A 2-SUBSTITUTED-INDOLE-1-LOWER-ALKANECARBOXAMIDES HAVING ANTI-SECRETORY OR ANTI-ULCER ACTIVITY STERLING DRUG INC. (US) 1978-01-17 US disclosed
US-4021448-A ANTISECRETORY AND ANTIULCER ACTIVITIES STERLING DRUG INC. (US) 1977-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12371429-B2 Antibiotic resistance-modifying tricyclic heteroaryl compounds and uses thereof CBR3, CBR1, CYP2B6 LMNA 2789/4885HPGD 3554/4885CYP1A2 233/4885
US-20210163479-A1 1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOLE DERIVATIVE COMPOUNDS AND USES THEREOF H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CCNA1, FOXM1 LMNA 1737/4885HPGD 2568/4885CYP1A2 578/4885
US-20100168417-A1 2-Indolyl Imidazo [4,5-d] Phenanthroline Derivatives and Their Use in the Treatment for Cancer FLI1, IKZF3, IKZF2 LMNA 1875/4885HPGD 1132/4885CYP1A2 1955/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.