SCHEMBL10243447

SCHEMBL10243447

CCN(CCNC(=O)OC)Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
APP P05067 3/20 0.54
OPRM1 P35372 5/20 0.53
OPRK1 P41145 5/20 0.53
KDM4E B2RXH2 1/20 0.52
ACKR3 P25106 1/20 0.49
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
GAA P10253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13303073 0.87 TAAR1 (0.52) APPOPRM1OPRK1KDM4EACKR3
SCHEMBL10243111 0.86 POLB (0.46) APPOPRM1OPRK1KDM4EACHE
SCHEMBL10243109 0.84 CHRNB2 (0.48) GAA
SCHEMBL10243465 0.84 HDAC3 (0.47) APPOPRM1OPRK1KDM4EBCHE
SCHEMBL10243105 0.81 APP (0.61) APPBCHEACHE
SCHEMBL13303011 0.80 TAAR1 (0.48) APPOPRM1OPRK1KDM4EACKR3
SCHEMBL10243384 0.80 ALDH1A1 (0.49) KDM4EGAA
SCHEMBL10243171 0.79 KDM4E (0.49) APPOPRM1OPRK1KDM4EGAA
SCHEMBL13037027 0.79 EPHX1 (0.50) KDM4EACHE
SCHEMBL10243147 0.79 CDYL (0.49) APPKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281292-A1 10a-Azalide Compound IL17A, AZI2, HDAC9 APP 4678/4885OPRM1 4835/4885OPRK1 4818/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.