SCHEMBL10244079

SCHEMBL10244079

CCc1ccc(C(C)N(CC)CCNC(=O)OC)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
OPRK1 P41145 8/20 0.40
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PKM P14618 1/20 0.36
HTT P42858 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 1/20 0.35
GLA P06280 1/20 0.35
KMT2A Q03164 1/20 0.35
OPRM1 P35372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10243510 0.88 ALOX5 (0.40) ALDH1A1OPRK1LMNAL3MBTL1SMN1; SMN2
SCHEMBL10243491 0.87 MEN1 (0.45) ALDH1A1OPRK1L3MBTL1SMN1; SMN2GLA
SCHEMBL10243433 0.87 MAPT (0.43) MAPTL3MBTL1HTTSMN1; SMN2KMT2A
SCHEMBL10244037 0.87 CYP1A2 (0.46) ALDH1A1OPRK1HPGDSMN1; SMN2GLA
SCHEMBL10243623 0.87 HPGD (0.40) ALDH1A1LMNAHPGDMAPTHTT
SCHEMBL10243497 0.86 SLC22A1 (0.43) ALDH1A1LMNAHPGDSMN1; SMN2
SCHEMBL10243869 0.85 BCHE (0.37) ALDH1A1OPRK1
SCHEMBL10243580 0.85 ACACB (0.49) ALDH1A1LMNAHPGDSMN1; SMN2
SCHEMBL10244695 0.84 SMN1; SMN2 (0.41) ALDH1A1LMNAMAPTL3MBTL1SMN1; SMN2
SCHEMBL10243544 0.84 LMNA (0.43) OPRK1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281292-A1 10a-Azalide Compound IL17A, AZI2, HDAC9 ALDH1A1 1939/4885TDP1 2672/4885OPRK1 4818/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.