SCHEMBL10243544

SCHEMBL10243544

CCN(CCNC(=O)OC)C(C)c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.43
CYP2C9 P11712 2/20 0.43
TSHR P16473 2/20 0.43
ADRA2A P08913 1/20 0.43
CYP2D6 P10635 1/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
HTR2B P41595 1/20 0.43
STAT6 P42226 1/20 0.43
KCNH2 Q12809 1/20 0.43
BLM P54132 1/20 0.42
EPHX2 P34913 10/20 0.40
CTSK P43235 1/20 0.38
CCR5 P51681 1/20 0.36
OPRK1 P41145 2/20 0.36
CYP2C19 P33261 1/20 0.35
CYP2J2 P51589 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10243510 0.85 ALOX5 (0.40) LMNAOPRK1
SCHEMBL10243623 0.84 HPGD (0.40) LMNACYP2C9TSHRCYP2D6CYP2C19
SCHEMBL10243433 0.84 MAPT (0.43) CYP2C9CYP2D6CYP2C19
SCHEMBL10244037 0.84 CYP1A2 (0.46) CYP2D6OPRK1
SCHEMBL10243491 0.84 MEN1 (0.45) OPRK1
SCHEMBL10244079 0.84 ALDH1A1 (0.40) LMNATSHROPRK1
SCHEMBL10243497 0.83 SLC22A1 (0.43) LMNAADRA2ACYP2D6KCNH2
SCHEMBL10243802 0.82 MGLL (0.45) LMNA
SCHEMBL10243580 0.81 ACACB (0.49) LMNACYP2D6
SCHEMBL10244695 0.81 SMN1; SMN2 (0.41) LMNACYP2C9TSHRCYP2D6EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281292-A1 10a-Azalide Compound IL17A, AZI2, HDAC9 LMNA 1467/4885CYP2C9 395/4885TSHR 1567/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.