SCHEMBL1024672

SCHEMBL1024672

COc1ccc(-c2c(-c3c(F)cc(F)cc3F)c(Cl)nn2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.39
BACE1 P56817 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.36
SRC P12931 1/20 0.36
BRAF P15056 1/20 0.36
KDR P35968 1/20 0.36
ATM Q13315 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MAOA P21397 1/20 0.36
KDM1A O60341 1/20 0.35
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
THPO P40225 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1023575 0.93 L3MBTL1 (0.39) L3MBTL1BACE1POLBATMNPC1
SCHEMBL1023884 0.87 CYP1A2 (0.38) BACE1PTGS1PTGS2CYP1A2CYP3A4
SCHEMBL1025606 0.86 GRM5 (0.38) SRCBRAFKDRKDM5AKDM4C
SCHEMBL1023290 0.84 NR1H2 (0.36) PTGS2
SCHEMBL1026639 0.80 PDE10A (0.37) LMNANPC1RAB9AKDM1ACYP1A2
SCHEMBL1027586 0.79 GRM8 (0.36) BACE1LMNAKDM1APTGS2CYP1A2
SCHEMBL1023890 0.79 MEN1 (0.36) PTGS2CYP3A4CYP2C9CYP2C19
SCHEMBL3581885 0.77 NPC1 (0.44) POLBNPC1RAB9APTGS2TSHR
SCHEMBL1026094 0.77 PDE10A (0.39) PTGS1PTGS2
SCHEMBL1025108 0.77 PDE10A (0.37) PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274285-A1 NOVEL PYRAZOLE DERIVATIVES Syngenta Participations AG (CH) 2011-01-19 EP claimed
WO-2009127612-A1 NOVEL PYRAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2009-10-22 WO claimed
EP-2274285-A1 NOVEL PYRAZOLE DERIVATIVES Syngenta Participations AG (CH) 2011-01-19 EP disclosed
WO-2009127612-A1 NOVEL PYRAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2009-10-22 WO disclosed