SCHEMBL1027586

SCHEMBL1027586

COc1cc(F)c(-c2c(Cl)nn(C)c2-c2ccc(C)nc2)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM8 O00222 1/20 0.36
CYP1A2 P05177 1/20 0.36
GRM7 Q14831 1/20 0.36
PDE10A Q9Y233 3/20 0.34
ABL1 P00519 1/20 0.34
BCR P11274 1/20 0.34
MAOB P27338 2/20 0.33
PDE2A O00408 2/20 0.33
BACE1 P56817 1/20 0.33
PTGS2 P35354 2/20 0.33
TP53 P04637 1/20 0.33
CTSA P10619 1/20 0.32
LMNA P02545 1/20 0.32
KDM1A O60341 1/20 0.32
IGF1R P08069 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1026639 0.89 PDE10A (0.37) GRM8CYP1A2GRM7PDE10AMAOB
SCHEMBL1025108 0.86 PDE10A (0.37) PDE10APDE2APTGS2TP53IGF1R
SCHEMBL1023575 0.85 L3MBTL1 (0.39) GRM8CYP1A2GRM7PDE10ABACE1
SCHEMBL1025104 0.84 PDE10A (0.36) PDE10AMAOBLMNA
SCHEMBL1023884 0.84 CYP1A2 (0.38) GRM8CYP1A2GRM7PDE10APDE2A
SCHEMBL1024672 0.79 L3MBTL1 (0.39) CYP1A2BACE1PTGS2LMNAKDM1A
SCHEMBL1026094 0.77 PDE10A (0.39) PDE10APDE2APTGS2TP53IGF1R
SCHEMBL1023890 0.77 MEN1 (0.36) PDE10APTGS2
SCHEMBL19953206 0.75 POLB (0.38) CYP1A2PDE10ABACE1PTGS2
SCHEMBL1025996 0.73 PDE10A (0.35) PDE10APDE2ATP53IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274285-A1 NOVEL PYRAZOLE DERIVATIVES Syngenta Participations AG (CH) 2011-01-19 EP claimed
WO-2009127612-A1 NOVEL PYRAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2009-10-22 WO claimed
EP-2274285-A1 NOVEL PYRAZOLE DERIVATIVES Syngenta Participations AG (CH) 2011-01-19 EP disclosed
WO-2009127612-A1 NOVEL PYRAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2009-10-22 WO disclosed