SCHEMBL10246754

SCHEMBL10246754

C=C(C)CN1CCCNCC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 12/20 0.47
SIGMAR1 Q99720 5/20 0.45
CHRM5 P08912 2/20 0.44
CHRM3 P20309 2/20 0.44
MEN1 O00255 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
ADRA2C P18825 1/20 0.42
CCR2 P41597 1/20 0.42
CXCL12 P48061 1/20 0.42
BLM P54132 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1126801 0.92 CHRM5 (0.46) CXCR4SIGMAR1CHRM5CHRM3
SCHEMBL28170665 0.83 CXCR4 (0.50) CXCR4SIGMAR1CHRM5CHRM3MEN1
SCHEMBL6826228 0.82 SIGMAR1 (0.48) CXCR4SIGMAR1CHRM5CHRM3MEN1
SCHEMBL8732181 0.80
SCHEMBL10248697 0.80
SCHEMBL12226505 0.80 CHRM5 (0.53) CXCR4SIGMAR1CHRM5CHRM3MEN1
SCHEMBL10283313 0.80 ALDH1A1 (0.58) CXCR4SIGMAR1CHRM5CHRM3MEN1
SCHEMBL9059440 0.79
SCHEMBL10246527 0.78 ALDH1A1 (0.45) MEN1KMT2ATDP1HRH3
SCHEMBL10248708 0.78 ALDH1A1 (0.45) MEN1KMT2ATDP1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120041193-A1 SUBSTITUTED INTERNAL VINYL-BORONIC ACIDS AND BORONIC ACID DERIVATIVES FRONTIER SCIENTIFIC, INC. (US) 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120041193-A1 SUBSTITUTED INTERNAL VINYL-BORONIC ACIDS AND BORONIC ACID DERIVATIVES BLVRB, BTD, BCL6B CXCR4 1349/4885SIGMAR1 4074/4885CHRM5 4642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.