SCHEMBL10246887

SCHEMBL10246887

CN(Cc1ccc(F)cc1)Cc1cc(CO)cc(-c2ccc(F)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 2/20 0.53
MCHR1 Q99705 4/20 0.41
NPC1 O15118 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
CSF1R P07333 1/20 0.39
PTGS1 P23219 1/20 0.39
KCNH2 Q12809 2/20 0.38
HTR2C P28335 1/20 0.38
GRM2 Q14416 1/20 0.38
ALOX5 P09917 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
CXCR3 P49682 1/20 0.37
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
RIPK1 Q13546 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22304838 0.83 PYCR1 (0.60) PYCR1NPC1CXCR3MEN1RAB9A
SCHEMBL19300926 0.79 PTGS1 (0.46) PTGS1RXRARXRBRXRG
SCHEMBL15164028 0.77 RXRA (0.44) PYCR1MCHR1PTGS1KCNH2HTR2C
SCHEMBL3191532 0.77 PYCR1 (0.67) PYCR1NPC1HRH3CXCR3MEN1
SCHEMBL30093198 0.77 PYCR1 (0.67) PYCR1NPC1HRH3CXCR3MEN1
SCHEMBL185132 0.74 LMNA (0.49) MCHR1PTGS1RXRARXRBRXRG
SCHEMBL4412749 0.73 PTGS1 (0.60) PYCR1PTGS1MEN1KMT2A
SCHEMBL27825225 0.72 HRH3 (0.77) PYCR1MCHR1HRH3ALOX5RIPK1
SCHEMBL3582959 0.71 PTGS1 (0.40) PTGS1RXRARXRBRXRGMEN1
SCHEMBL3591800 0.71 AGXT (0.41) PTGS1RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297103-B1 HYDROXYPHENYLSULFONAMIDES AS ANTIAPOPTOTIC BCL INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2012-01-04 EP disclosed