SCHEMBL10248596

SCHEMBL10248596

COC(=O)CN1C(=O)[C@@H](NBC=O)CNc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
XIAP P98170 2/20 0.43
PYGL P06737 1/20 0.39
LMNA P02545 1/20 0.38
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.37
SCN9A Q15858 1/20 0.36
POLB P06746 1/20 0.36
RIPK1 Q13546 2/20 0.36
OPRL1 P41146 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13139827 0.82 XIAP (0.47) XIAPPYGLLMNAALDH1A1SCN9A
SCHEMBL14370029 0.81 XIAP (0.42) XIAPPYGLLMNAALDH1A1SCN9A
SCHEMBL645568 0.80 SCN9A (0.51) XIAPSCN9A
SCHEMBL645694 0.80 SCN9A (0.51) XIAPSCN9A
SCHEMBL4556966 0.80 NAAA (0.47) XIAPPYGLLMNASCN9AOPRL1
SCHEMBL648535 0.80 XIAP (0.48) XIAPPYGLALDH1A1RIPK1MEN1
SCHEMBL14370027 0.80 XIAP (0.42) XIAPPYGLLMNAALDH1A1POLB
SCHEMBL645717 0.79 LMNA (0.43) XIAPPYGLLMNAALDH1A1POLB
Hydrochloric Acid SCHEMBL645716 0.78 LMNA (0.42) XIAPPYGLLMNAALDH1A1POLB
SCHEMBL645689 0.77 RIPK1 (0.44) XIAPPYGLRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119631-B2 Inhibitors of interleukin-1β converting enzyme VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-21 US disclosed