SCHEMBL10249655

SCHEMBL10249655

CC(=O)C[C@@H](C=O)NC(=O)CN1C(=O)[C@@H](NC(=O)/C=C/c2ccccc2)CN(C(C)=O)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
XIAP P98170 15/20 0.41
MMP2 P08253 2/20 0.41
ANPEP P15144 1/20 0.41
CYP3A4 P08684 8/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
TP53 P04637 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10199339 0.95 XIAP (0.41) XIAPMMP2ANPEPCYP3A4SMN1; SMN2
SCHEMBL10200499 0.90 XIAP (0.38) XIAPCYP3A4SMN1; SMN2
SCHEMBL13139782 0.89 MAPT (0.40) XIAPSMN1; SMN2TP53ALDH1A1
SCHEMBL10200507 0.89 MAPT (0.40) XIAPSMN1; SMN2TP53ALDH1A1
SCHEMBL10249823 0.86 CASP1 (0.47) XIAPCYP3A4
SCHEMBL10249657 0.86 XIAP (0.46) XIAPCYP3A4
SCHEMBL10201832 0.85 MAOB (0.40) XIAPSMN1; SMN2TP53ALDH1A1
SCHEMBL10199522 0.85 XIAP (0.42) XIAPCYP3A4
SCHEMBL10249659 0.83 CASP1 (0.47) XIAPCYP3A4
SCHEMBL644702 0.81 CASP1 (0.47) XIAPCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119631-B2 Inhibitors of interleukin-1β converting enzyme VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-21 US disclosed
US-20110178069-A1 INHIBITORS OF INTERLEUKIN-1 BETA CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-07-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178069-A1 INHIBITORS OF INTERLEUKIN-1 BETA CONVERTING ENZYME IL1A, IFNAR1, IL1B XIAP 257/4885MMP2 317/4885ANPEP 82/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.