SCHEMBL1025879

SCHEMBL1025879

CC(C)(C)N(C(=O)O)c1ccnc(CCc2cccc(Nc3nc(Cl)ncc3F)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
SYK P43405 5/20 0.41
EGFR P00533 9/20 0.38
ITK Q08881 6/20 0.38
BTK Q06187 1/20 0.38
CCNT1 O60563 3/20 0.38
CDK9 P50750 3/20 0.38
CCNE1 P24864 2/20 0.38
CDK2 P24941 2/20 0.38
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1023949 0.92 ALDH1A1 (0.40) ALDH1A1EGFRBTKKDM4EGAA
SCHEMBL1026292 0.87 SYK (0.42) ALDH1A1SYKEGFRITKBTK
SCHEMBL1026319 0.86 SYK (0.42) ALDH1A1SYKEGFRITKBTK
SCHEMBL1025701 0.83 ALDH1A1 (0.49) ALDH1A1SYKEGFRITKBTK
SCHEMBL13623035 0.82 SYK (0.55) ALDH1A1SYKEGFRITKCCNT1
SCHEMBL13623036 0.79 SYK (0.48) ALDH1A1SYKEGFRITKBTK
SCHEMBL4328037 0.79 NR3C2 (0.47) ALDH1A1SYKEGFRITKBTK
SCHEMBL1025143 0.78 BCL6 (0.40) ALDH1A1SYKEGFRITKBTK
SCHEMBL1027536 0.78 SYK (0.44) SYKEGFRITKBTKCCNT1
Hydrochloric Acid SCHEMBL1026587 0.78 SYK (0.47) ALDH1A1SYKEGFRITKBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274288-A2 MACROCYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS Incyte Corporation (US) 2011-01-19 EP disclosed