SCHEMBL1023949

SCHEMBL1023949

CC(C)(C)N(C(=O)O)c1ccnc(CCc2cccc(Nc3nc(Cl)ncc3Cl)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
BCL6 P41182 1/20 0.38
CTSC P53634 2/20 0.37
BTK Q06187 2/20 0.36
EGFR P00533 7/20 0.35
HSD11B1 P28845 1/20 0.35
KDR P35968 3/20 0.35
JAK3 P52333 3/20 0.34
RHOA P61586 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1025879 0.92 ALDH1A1 (0.43) ALDH1A1KDM4EGAABTKEGFR
SCHEMBL1025143 0.87 BCL6 (0.40) ALDH1A1BCL6CTSCBTKEGFR
SCHEMBL1026953 0.84 GAA (0.47) ALDH1A1GAABCL6BTK
SCHEMBL1027670 0.84 BCL6 (0.38) ALDH1A1BCL6CTSCBTKEGFR
SCHEMBL1026721 0.83 JAK3 (0.42) BCL6CTSCJAK3
SCHEMBL1026395 0.83 BCL6 (0.40) BCL6CTSCBTKEGFRJAK3
SCHEMBL4348221 0.83 ALDH1A1 (0.46) ALDH1A1KDM4EGAACTSCBTK
SCHEMBL1023285 0.82 ALK (0.40) ALDH1A1BCL6BTK
SCHEMBL1025086 0.81 BCL6 (0.38) ALDH1A1BCL6CTSCBTKEGFR
SCHEMBL13623027 0.81 SYK (0.44) ALDH1A1KDM4EGAABCL6BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274288-A2 MACROCYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS Incyte Corporation (US) 2011-01-19 EP disclosed